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8-(5-phenoxyfuran-2-carbonyl)-1-oxa-8-azaspiro[4.5]decane
2-(piperidine-1-carbonyl)-6-{pyrazolo[1,5-a]pyridin-7-yl}pyrazine
2-hydroxy-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
N-(butan-2-yl)-6-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazine
4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-1-carboxamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(propan-2-yl)urea
N-(2-cycloheptylethyl)-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
2-[2-methyl-4-(1-methyl-1H-pyrazol-4-yl)phenoxy]acetamide
2-(2,4-dimethoxyphenyl)-2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]acetic acid
N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-cyclopentanecarbonyl-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
2-(3-fluoro-4-methoxyphenyl)-2-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}acetic acid
5-{[4-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-ethyl-4-methyl-1H-imidazole
N-[(3,4-difluorophenyl)methyl]-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]propanamide
(2-{2-[1-(6-chloroquinolin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
5-ethyl-1'-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(6-chloro-2-methylpyridin-3-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
1-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
1-(2-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
2-[3-(4-fluorophenyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzoic acid
methyl 2-{[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl](methyl)amino}acetate
{[3-chloro-5-ethoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}[1-(1-methyl-1H-pyrazol-5-yl)propyl]amine
N-[3-(2-amino-6-fluoro-1,3-benzothiazol-4-yl)phenyl]acetamide
8-[(2,6-difluorophenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
butyl 3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxylate
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(4-methylphenyl)sulfanyl]piperidine
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
2-(2-methoxy-5-methylphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
3-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}phenol
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)naphthalene-1-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
N3-benzyl-1-cyclohexyl-N5-cyclopropyl-N3-(2-hydroxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{[1-(2,2-dimethylpropanoyl)piperidin-3-yl]methyl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
(4S,4aS,8aS)-1-(cyclopropanesulfonyl)-4-phenyl-decahydroquinolin-4-ol
8-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(4aR,8aR)-2-(2-aminopyrimidin-4-yl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-propyl-1,3-thiazole-4-carboxamide
2,8-dimethyl-4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)quinoline
3,5-dimethyl-4-[1-(1,3-thiazol-4-ylmethyl)pyrrolidin-2-yl]-1,2-oxazole
1-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
2,5-dimethoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(piperidin-1-yl)ethyl]acetamide
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
8-[(2,5-difluorophenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
7-methyl-6-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one