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2-(2-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}phenoxy)acetamide
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
(1S,5R)-3-(3-phenylpropyl)-6-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[1-(2-ethylbutyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
4-[2-(dimethylamino)ethyl]-1-(2,6-dimethylpyridine-4-carbonyl)-1,4-diazepan-5-one
2-hydroxy-5-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)benzoic acid
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
5-({5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2-methylphenol
4-cyclopentyl-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]pyrimidin-2-amine
(3aS,7aR)-2-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
N-[(1R,3R)-3-aminocyclopentyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
7-fluoro-2-methyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}quinoline
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
3-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[2-(piperidin-1-ylmethyl)phenyl]urea
N,1-diethyl-5-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
1-(2,6-dimethylpyridin-4-yl)-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazine
N-cyclopropyl-2-ethyl-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}butanamide
3-(1-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-(2,8-dimethylquinoline-4-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-(2-phenylethyl)-8-{[4-(propan-2-yl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-1,4-diazepan-6-ol
4-({4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)benzonitrile
4-[(2S)-1-[4-(1H-pyrazol-1-yl)benzoyl]pyrrolidine-2-carbonyl]morpholine
1-({4-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)-4-methylpiperidine-4-carbonitrile
N-[(4-fluorophenyl)methyl]-3-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]propanamide
2-[(2-ethylpiperidin-1-yl)methyl]-4-(pyrimidin-2-yl)phenol
4-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-4-oxobutane-1-sulfonamide
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{[4-(methylsulfanyl)phenyl]methyl}-1,3-oxazole-4-carboxamide
7-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
(3S,9aR)-8-benzoyl-3-ethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-hydroxyethyl)-N-(propan-2-yl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[3-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-amino-1-(4-{[5-(hydroxymethyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-methylpropan-1-one
N-cyclopentyl-4-[(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(2-fluorophenyl)methyl]-1H-pyrazole-3-carboxamide
3-(diethylamino)-1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}propan-1-one
(2R)-1-({4-[(2-propyl-2H-1,2,3-triazol-4-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)oxane-4-carboxamide
3-(2-methoxyethyl)-5-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazole
3-fluoro-5-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]benzonitrile
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)acetamide
N,1,3-trimethyl-N-{1-[1-(3-methylbutyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-5-carboxamide
2-(4-chloro-1H-pyrazol-1-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
(1S,2R)-1-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]-2,3-dihydro-1H-inden-2-ol
3-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione