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N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-N,2,2,6,6-pentamethylpiperidin-4-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridine-2-sulfonyl)ethyl]amine
5-(1H-imidazol-1-ylmethyl)-2-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyridine
1-{4-[(2-hydroxyethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
5-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
(1S,3R)-3-amino-N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)cyclopentane-1-carboxamide
6-(3-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-3-oxopropyl)-2,3,4,5-tetrahydropyridazin-3-one
2-{[(3R,5S)-1-[(2,5-difluorophenyl)methyl]-5-(morpholine-4-carbonyl)pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-[2-(1H-pyrrol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,4R)-4-ethyl-1-(2-methyl-1-benzofuran-7-carbonyl)piperidine-3,4-diol
(3aS,6aS)-2-[2-chloro-5-(trifluoromethyl)benzoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2-dimethylthieno[3,2-d]pyrimidin-4-amine
[7-(2,6-dimethylpyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-7-acetamido-1-[(4-fluorophenyl)methyl]-N-methyl-1H-1,3-benzodiazole-5-carboxamide
2-[5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
1-(2-methylpropyl)-4-[2-(morpholin-4-yl)pyridin-3-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
4-{3-[(3-chlorophenyl)methyl]-5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
dimethyl(2-{1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-2-yl}ethyl)amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
9-(2-amino-6-methoxypyrimidin-4-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-acetamido-N,N-diethyl-1-[(5-fluoro-2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-amino-1-{[4-(2-methylphenyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl 2-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methylacetamido]acetate
ethyl 1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
2-(3-chloro-4-fluorophenyl)-4-(pyrrolidine-1-carbonyl)pyridine
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-(1-methylpiperidin-4-yl)piperidine
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-ethyl-1H-1,2,4-triazole
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(5-methylfuran-2-yl)-N-propyl-1H-pyrazole-5-carboxamide
4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(5-{[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-3-yl)pyridine
4-(dimethylamino)-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
1-(2-chlorophenyl)-4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
N-methyl-N-[1-(pyridin-3-yl)pentyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
6-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
methyl 4-{2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamido}butanoate
6-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carboxylic acid
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-{4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazin-1-yl}pyrimidine
3-(4-{[2-(difluoromethoxy)phenyl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
2-({[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
9-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
N-(2,2-difluoroethyl)-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}benzamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(1-methylazepane-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate