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N-[2-(1-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperidin-2-yl)ethyl]acetamide
N-{2-[4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3-methylpyridin-2-amine
{2-methyl-3-[2-(2,4,6-trifluorophenyl)-1H-imidazol-1-yl]phenyl}methanol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
1-[(5-methylfuran-2-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-[2-(2,6-difluorophenyl)ethyl]-1-(dimethyl-1,3-oxazole-4-carbonyl)piperidine
4-{[3-(2-methyl-1,3-thiazol-4-yl)-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
4,5-dimethyl-6-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
N-{2-[2-(6-methylquinolin-5-yl)-1H-imidazol-1-yl]ethyl}acetamide
2-amino-1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
5-(4-cyclopentylpiperazin-1-yl)-N-[(2-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{4-[3-phenyl-5-(thiomorpholine-4-sulfonyl)benzoyl]piperazin-1-yl}ethan-1-ol
1-methyl-6-oxo-N-[2-(3-phenoxyphenyl)ethyl]piperidine-3-carboxamide
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-3-ol
4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1H-pyrrole-2-carbonyl)piperidine
3-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(3R,4R)-1-{[4-(benzyloxy)phenyl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
N-cyclopropyl-3-(3-fluorophenyl)-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)benzamide
N-[(3R,4S)-1-[3-(4-fluorophenyl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
4-methyl-N-{2-[7-(3-methylbut-2-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[3-(1H-1,2,4-triazol-5-yl)phenyl]methyl}amine
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3-carboxamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-2-methyl-1H-1,3-benzodiazole-5-carboxamide
3-(azepane-1-carbonyl)-N-[2-(2-methoxyphenyl)ethyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 4-{[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-pyrazole-3-carboxylate
(2R,6S)-4-[6-chloro-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]-2,6-dimethylmorpholine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
N-(2-phenylethyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
2-{4-[(4-fluorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
(2S)-N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
1-{2-[(2-amino-5-butyl-6-methylpyrimidin-4-yl)amino]ethyl}piperidin-4-ol
(1S,5R)-3-[2-(2,4-dichlorophenoxy)acetyl]-3,9-diazabicyclo[3.3.2]decan-10-one
5-({[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(pyridin-3-yl)spiro[2.4]heptane-1-carboxamide
1-{[4-(difluoromethoxy)phenyl]methyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
methyl 2-(benzylsulfamoyl)-6-[(2,4-difluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl[(1-methyl-1H-imidazol-2-yl)methyl]{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
(4aR,8aS)-1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-6-(furan-2-carbonyl)-decahydro-1,6-naphthyridine
4-[(2,5-difluorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
N-[(2-methylphenyl)(phenyl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2,5-dimethyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
(3S,4S)-4-(morpholin-4-yl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidin-3-ol
N4-(2,1,3-benzothiadiazol-5-ylmethyl)-N4,6-dimethylpyrimidine-2,4-diamine