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5-methyl-1-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
[4-({1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-(6-aminopyrimidin-4-yl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
3-(3-chloro-1,2-oxazol-5-yl)-N-[2-(2-ethoxyphenoxy)ethyl]-N-methylpropanamide
(1R,2S,6R,7S)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-4-azatricyclo[5.2.2.02,6]undecane
2-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}-N-(thiophen-2-ylmethyl)quinazolin-4-amine
1'-(1-benzofuran-5-ylmethyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-({2-[1-(5-ethylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-3-phenylpiperazine
6-(2,3-dimethoxyphenyl)-N,N-dimethylpyridine-2-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-4-(piperidin-1-yl)butanamide
1-{1-[3-(4-methylphenyl)phenyl]piperidin-4-yl}piperidine-4-carboxamide
N-(3-cyclopentylpropyl)-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(2-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}phenoxy)acetamide
3-methyl-6-(3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridazine
(1R,2S)-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-2-propylcyclopropane-1-carboxamide
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-(oxan-4-yl)-3-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
2-(4-fluorophenyl)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]azetidine
ethyl 1-(pyridin-2-ylmethyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-[2-(5-acetylthiophen-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-4-(trifluoromethyl)benzamide
N,N-dimethyl-4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}aniline
3-[3-(2-chlorophenyl)pyrrolidin-1-yl]-5-(4-methoxyphenyl)-1,2,4-triazine
4,6-dimethyl-1-[2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]-1,2-dihydropyrimidin-2-one
N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)cyclopropanesulfonamide
N-(4-methoxy-2-methylphenyl)-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
methyl 5-[(3-hydroxybutyl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
5-[(methylsulfanyl)methyl]-N-[1-(pyridine-3-carbonyl)azepan-3-yl]furan-2-carboxamide
1-(4-methoxyphenyl)-2-[1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
(2R,3R,6R)-5-(2,3-dihydro-1-benzofuran-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3aR,6aR)-2-(2-aminopyrimidin-4-yl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(4-methoxyphenyl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
methyl 2-[1-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazol-4-yl)-N-methylformamido]acetate
(3R,4R)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
4-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
4-methyl-1-(2-{2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-1H-1,2,3-triazole
N-{[7-(1H-indole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-methylthiophene-2-carboxamide
N-(2-{1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-2-yl}ethyl)acetamide
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-(4-phenylbutanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(3S,4R)-1-(3-hydroxy-4-methoxybenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
5-(azepane-1-carbonyl)-1-[2-(4-chlorophenyl)ethyl]piperidin-2-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-4-[(2-hydroxyethyl)(methyl)amino]benzamide
1-(4-{4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)-3-(1H-pyrrol-1-yl)propan-1-one
2-[4-(1-benzofuran-2-ylmethyl)-1-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
2-chloro-5-{[(oxan-3-ylmethyl)carbamoyl]amino}-N-propylbenzamide