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(1S,5R)-6-benzyl-3-(4-chloro-2-hydroxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{4-[(3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-phenylpropan-1-ol
1-[2-(3-ethoxyphenyl)pyridine-4-carbonyl]-4-methylpiperazine
(2E)-3-(2-fluorophenyl)-1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)prop-2-en-1-one
3-{1-[3-(3,5-dimethylphenyl)propanoyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]acetamide
3-[(4-fluorophenyl)formamido]-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)propanamide
ethyl 1-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)piperidine-3-carboxylate
(2R,6R)-4-(4-oxo-4-phenylbutyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-{[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}-N-(1,3-thiazol-2-yl)propanamide
2-(azonan-1-yl)-7-methanesulfonyl-4-methylquinazoline
[2-(quinolin-8-yl)quinolin-3-yl]methanol
N-tert-butyl-2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}acetamide
N-cyclopropyl-1-[1-(1-methylazepane-2-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
2-methyl-6-[(6-methylhept-5-en-2-yl)amino]heptan-2-ol
1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-[4-({4-[2,5-dioxo-4-(3-phenylpropyl)imidazolidin-4-yl]piperidin-1-yl}methyl)phenyl]acetamide
N-{[4-(morpholin-4-yl)phenyl]methyl}-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-{4-hydroxy-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-(3,3-dimethylbutanoyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
[(2-ethylpyrimidin-4-yl)methyl](methyl)[(1-phenylpyrrolidin-3-yl)methyl]amine
N-[1-(4-ethoxyphenyl)propyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-{4-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-ol
N-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}amine
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-[(3-methoxyphenyl)amino]butan-1-one
1-(azocan-1-yl)-3-(2-methoxy-4-{[(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
2-(4-chlorophenyl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-hydroxyacetamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]benzonitrile
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(furan-2-yl)-3-phenylpropan-1-one
(3R)-1-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
3-hydroxy-1-(3-phenylpropyl)-3-{[(prop-2-en-1-yl)amino]methyl}piperidin-2-one
(1R,3S)-3-ethoxy-7-[1-(2-methylphenyl)piperidin-4-yl]-7-azaspiro[3.5]nonan-1-ol
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N-phenylacetamide
N-[(3R,4S)-1-{2-[cyclopentyl(methyl)amino]acetyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-(2-chlorophenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylpropanamide
4-{1-[6-(3,4-dimethylpiperazin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
N,N-diethyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-benzyl-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1,3-thiazole-4-carboxamide
6-[2-(azepan-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyethyl)piperazine
4-benzyl-3-{1-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-ethyl-9-(6-methylpyrimidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine
3-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)pyrrolidin-2-yl]-5-methyl-1,2-oxazole