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1-(cyclohexylmethyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
1-{[4-(2-methylphenyl)phenyl]methyl}-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
methyl 3-{[(4-tert-butylphenyl)formamido]methyl}-5-(1,3-dimethyl-1H-pyrazole-5-amido)benzoate
2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
7-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2,4-difluorophenyl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
methyl 3-acetamido-5-{[(2-fluorophenyl)methyl]amino}-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
methyl 2-(cyclopropylsulfamoyl)-6-(naphthalen-1-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
1-[(3S)-3-(dimethylamino)azepan-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(4S)-3-(2-oxo-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-4-(propan-2-yl)-1,3-oxazolidin-2-one
2-{9-[2-(methylsulfanyl)propanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
2-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
5-(pyridin-4-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(4-phenyl-5-propyl-1H-imidazol-2-yl)pyrrolidin-2-one
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(2-hydroxybutyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-(1-ethyl-2-methyl-1H-indol-5-yl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carboxamide
1-{4-[(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)methyl]thiophen-2-yl}ethan-1-one
N-(1-methoxybutan-2-yl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
N-(6-hydroxy-6-methylheptan-2-yl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-(4-methoxybutyl)-N-{3-[(propan-2-yl)carbamoyl]phenyl}piperazine-1-carboxamide
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(thiophen-3-ylmethyl)piperidin-4-amine
N-[4-(1H-imidazol-1-yl)phenyl]-3-propoxypiperidine-1-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]quinoxaline-5-carboxamide
4-[(2-methoxyphenyl)methyl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
2-(pyridin-3-yl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrimidine-5-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(hydroxymethyl)cycloheptyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
ethyl (4aS,8aR)-6-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-decahydro-1,6-naphthyridine-4a-carboxylate
1-methyl-N-(1,3,4-thiadiazol-2-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carboxamide
6-[(2-methoxyethyl)(methyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-methyl-4-[1-(4-phenylbenzoyl)pyrrolidin-3-yl]piperazine
{4-[(2-chlorophenyl)methyl]-1-phenylmethanesulfonylpiperidin-4-yl}methanol
N-[3-fluoro-5-(trifluoromethyl)phenyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
(2S,4R)-4-amino-1-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-methoxy-4-methyl-N-[(1-methylpiperidin-4-yl)methyl]benzamide
8-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{2-[4-(3-chloro-5-methylpyridin-2-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(methoxymethyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-[(4-fluorophenyl)methyl]-5-(1-methylpyrrolidin-3-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-[2-(1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
2-{1'-[(3-methoxyphenyl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
3-(2-ethyl-1H-imidazol-1-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylpropanamide
2-acetyl-8-(4-propoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane