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4-[3-(piperidin-4-ylmethyl)benzoyl]-1λ6-thiomorpholine-1,1-dione
6-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyrimidin-4-amine
2-(4-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)pyridine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,3-dimethylthiophene-2-carboxamide
1-methyl-2-{5-phenyl-1H-pyrazolo[3,4-b]pyridin-6-yl}-1H-imidazole
9-(3,5-dimethylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(4-methylphenyl)methyl]-1H-pyrazole-4-carboxamide
methyl 8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1-methyl-N-(2-phenylethyl)piperidin-4-amine
N-[7-(4-acetylpiperazine-1-carbonyl)-1-(2-methoxyethyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
2-(1-{2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazol-4-yl}-N-methylformamido)-N-methylacetamide
N-[1-(4-fluorophenyl)ethyl]-3-(2-methyl-5-oxopyrrolidin-2-yl)propanamide
2-(2-methoxyethyl)-5-{1-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
3-[(3R,4S)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
6-(methoxymethyl)-N,1-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-2-phenyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
4-[4-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)phenyl]-2-methylbutan-2-ol
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[3-(morpholin-4-yl)propyl]amine
2-[4-(isoquinolin-5-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
1-cyclohexyl-4-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine
4-[4-(3,4-difluorophenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[2-(oxan-2-yl)ethyl]acetamide
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-(ethylsulfanyl)pyrimidine
N3-(1-benzylpiperidin-4-yl)-1-cyclopentyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-1-benzofuran-5-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-one
1-(carbamoylmethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
2-{5-[5-(methoxymethyl)furan-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
6-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)naphthalen-2-ol
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2,2-diphenylacetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
(4aR,7aS)-1-ethyl-4-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-N-[(3-methylthiophen-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
(3S,9aR)-3-(4-aminobutyl)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-6-[2-(methylamino)pyridine-4-carbonyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]oxane-4-carbonitrile
3-(1H-imidazol-1-yl)-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(piperidine-1-carbonyl)piperidine
8-(4-methyl-1H-pyrrole-2-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(7-{[4-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-4-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}methanesulfonamide
(2R)-N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrrolidine-2-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-[1-(pyridin-3-yl)pentyl]acetamide
(3S,4R)-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
(3S,7S)-5-[2-(methylamino)-1,3-thiazole-4-carbonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid