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3-(3-methoxypropyl)-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
N-[2-(dimethylamino)ethyl]-6-ethyl-N-(2-hydroxyethyl)-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
5-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
7-(4-chlorophenyl)-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)azepan-4-ol
1-ethyl-3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}-1-(oxan-2-ylmethyl)urea
2,5-dimethyl-3-{4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}pyrazine
3-(1H-imidazol-2-yl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidine
8-(1,3-benzothiazol-2-yl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-ethyl-2-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1,3-thiazole-5-carboxamide
(4aS,7aR)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-fluoro-2-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine-4-carboxylate
methyl 2-[N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]acetate
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2,5-dimethoxyphenyl)-N-{[7-fluoro-2-(thiophen-2-yl)quinolin-3-yl]methyl}acetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}propan-1-one
4-(4-methylphenyl)-3-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-2-(1H-1,2,4-triazol-3-yl)benzamide
2-fluoro-N-methyl-N-(1,2-oxazol-5-ylmethyl)-5-sulfamoylbenzamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(1H-pyrazol-1-yl)butan-1-one
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[(3S,4R)-1-(5-chloro-2-methoxybenzoyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
methyl (2S,4R)-4-(2-phenylbenzamido)-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)cyclohexanecarboxamide
N-(1-phenylbutyl)furan-2-carboxamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-hydroxy-3-methylbenzamide
5-methyl-5-(4-methylpent-3-en-1-yl)-1-{3-[(pyridin-3-yl)amino]propyl}piperidin-2-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(6-methylpyridine-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-methoxy-2-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-4H-pyran-4-one
3-(3,4-dimethoxybenzoyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
N-(1-benzothiophen-2-ylmethyl)-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-methylacetamide
1-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-yl}-2-phenylethan-1-one
2-methyl-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-(1-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-4-(1H-pyrazol-3-yl)benzamide
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N-butyl-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-(2-methoxyphenoxy)-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
2-[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-cyclopropyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[(2-methoxyphenyl)methyl]acetamide
2-[(4aR,7aS)-4-(cyclobutylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[(3S,4R)-4-(4-methylphenyl)-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-3-yl]acetamide
N-cyclopentyl-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
butyl (1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate