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3-{[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]sulfonyl}-N-(2-fluoroethyl)benzamide
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
(2E)-4-methyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-2-enamide
N3-ethyl-N5-[2-(3-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(3-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl]amino}phenyl)-N-methylacetamide
2-[4-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
2-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}pyridine
N-ethyl-5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-amine
(2S,4R)-N-methyl-4-[4-(2-{[(2-methylphenyl)carbamoyl]amino}propan-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}cyclopropane-1-carbonitrile
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N,1,3,6-tetramethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1H-indazole-3-carboxamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-(propan-2-yl)urea
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
N-[3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)carbamoyl}amino)-4-methoxyphenyl]acetamide
3,8-dibenzyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-benzyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,3-thiazole-4-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-ethyl-2-methylpyrimidine
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(1-{[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3,5-dichloro-4-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}benzamide
N-[2-(3-ethoxyphenoxy)ethyl]-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
[(1S,3S,3aS,6aR)-5-ethyl-3-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-1,4-diazepane-6-carboxylic acid
3-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
6-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]pyridine-3-carboxylic acid
2-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}sulfonyl)benzonitrile
2-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2-methylphenyl)-4-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)piperazine
3-{2-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
1-(4-{[4-(prop-2-yn-1-yloxy)phenyl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecan-11-yl)propan-1-one
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
4-(1H-imidazol-2-yl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]prop-2-en-1-one
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-5-oxopyrrolidine-2-carboxamide
{5-fluoro-7-[2-(piperazin-1-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-{4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazin-1-yl}pyrimidine
1-[4-(5-aminopyridin-3-yl)phenyl]cyclopentane-1-carbonitrile
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-1H-pyrazole-4-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
2-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}benzonitrile
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
3-(2-methoxyphenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]benzamide
3-(1-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazol-4-yl)phenol