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5-{[(7-chloroquinolin-4-yl)amino]methyl}pyrrolidin-2-one
(3R,9aR)-8-[(3-chlorophenyl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-oxobutanamide
4-[3-(pyridin-4-yl)azetidin-1-yl]-8-(trifluoromethyl)quinoline
N6-(3-methoxypropyl)-N5-methyl-N5-[(1-methylpiperidin-2-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-benzyl-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,3-benzoxazole-5-carboxamide
2-{5-[(1R,2R)-1-amino-2-hydroxypropyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-butyl-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
methyl 3-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanoate
4-chloro-2-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}phenol
ethyl 4-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
5-methyl-N-[2-(quinolin-8-yloxy)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[5-(butoxymethyl)-3-methyl-1H-1,2,4-triazol-1-yl]-6-methylpyridine
4-(3-methylphenoxy)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylic acid
5-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[3-(4-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(1H-indazol-1-yl)acetamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
8-(3-hydroxybenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 4-(6-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
2-(dimethylamino)-1-[4-(3-methoxypropyl)piperidin-1-yl]-2-(2-methylphenyl)ethan-1-one
2-(ethylamino)-N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
N3-ethyl-4-oxo-1-(2-phenylethyl)-N5-{[2-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-methyl-1,2-oxazole-3-carboxamide
5-benzamido-1-cyclopentyl-N-(1-methoxybutan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
1-cyclopropyl-4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
(4aS,8aR)-6-[(4-methyl-1H-imidazol-5-yl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
2-(1-methyl-1H-pyrazol-4-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
3-[3-(3,4-dimethoxyphenyl)phenyl]-1-methyl-1H-pyrazole
1-ethyl-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]piperidin-2-one
5-(methoxymethyl)-N-({3-methyl-7-[3-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
6-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzothiazole
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-[(1-cycloheptylpiperidin-3-yl)carbamoyl]-2,1,3-benzoxadiazol-1-ium-1-olate
3-[(1-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
4-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-methyl-5-phenyl-1H-pyrazole
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoacetamide
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(4-fluorophenyl)methyl]methylamine
2-methoxy-1-[1'-(piperidin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2,5-dimethyl-N-[1-(pyridin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(1H-imidazol-2-yl)-1-methyl-1H-pyrazole
2-(dimethylamino)-N,4-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidine-5-carboxamide
3-({1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperidin-4-yl}methyl)benzoic acid
5-acetyl-3-(3-cyclopentyl-1-phenyl-1H-1,2,4-triazol-5-yl)-6-methyl-1,2-dihydropyridin-2-one
2-methyl-7-{[4-(methylsulfanyl)phenyl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide