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1-ethyl-N-[(6-methylquinolin-5-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1H-pyrazol-1-yl)propanamide
3-(3-hydroxyquinoxalin-2-yl)-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}propanamide
1-cyclopentyl-3-(3-fluorophenyl)-3-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione
N-(2-{[1-(furan-2-ylmethyl)piperidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
N-(3-fluoro-2-methylphenyl)-2-{[4-(pyrrolidin-1-yl)butyl]amino}acetamide
8-{[(3-fluorophenyl)methyl]carbamoyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{3-[3-(pyridin-3-yl)phenyl]-1H-pyrazol-1-yl}-N-(thiophen-2-ylmethyl)acetamide
N-[4-(3-acetamidophenyl)phenyl]-N-methylacetamide
1-(azocan-1-yl)-3-[2-methoxy-5-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N,2-dimethyl-N-(1,2-oxazol-3-ylmethyl)-6-(propan-2-yl)pyrimidin-4-amine
2-[1-cyclopentyl-4-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
N-(2-methoxyethyl)-1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(2-ethoxypyridin-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-({2-amino-6-[(propan-2-yl)amino]pyrimidin-4-yl}amino)ethyl]pyridine-4-carboxamide
3-(1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}piperidin-4-yl)-N-(3-methylphenyl)propanamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[3-(1H-pyrazol-1-yl)propyl]amine
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2,5-dimethoxybenzamide
({5-[1-(4-chlorobenzoyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
methyl 4-(4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
5-acetyl-N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2,4-dimethyl-1H-pyrrole-3-carboxamide
N,1-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[1-(2,5-dimethylphenyl)ethyl]-2-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
2-(dimethylamino)-N-[2-(2-hydroxyethoxy)ethyl]-2-(4-methylphenyl)acetamide
1-cycloheptanecarbonyl-4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine
2-{1-[(2-fluorophenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(3R,4S)-1-(1H-imidazole-2-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-amine
1-ethyl-2-{4-[1-(pyrimidin-2-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}-1H-1,3-benzodiazole
1-(2-methylphenyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
4-(1-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)morpholine
3-(azepane-1-carbonyl)-N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(6-aminopyridin-3-yl)phenyl]acetamide
2-methyl-2-[2-(4-methylpiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]propanoic acid
1-{[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-hydroxyazepan-4-yl]methyl}-3,3-dimethylurea
3-phenyl-N-(1-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
8-(3,5-difluoropyridine-2-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(quinolin-8-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-2-amino-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-hydroxypropan-1-one
1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
3-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)-N-(pyridin-3-yl)benzamide
2-{2-[(1-cyclopentylpiperidin-3-yl)formamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl})(pyrazin-2-ylmethyl)amine
6-{1-[(2,7-dimethyl-1H-indol-3-yl)methyl]piperidin-4-yl}-2-methyl-3,4-dihydropyrimidin-4-one
1-[3-(morpholin-4-yl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(oxolan-3-ylmethyl)piperidin-4-ol
5-acetyl-2,4-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrrole-3-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol