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2-cyclopentyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-phenylacetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-3-ol
methyl 4-methoxy-3-[(2-methyl-5-oxo-1,4-diazepane-1-carbonyl)amino]benzoate
methyl 3-acetamido-5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
N-cyclopentyl-3,5-dimethoxy-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzamide
N-benzyl-N-butyl-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)methylamine
3-({2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxypyrimidin-5-yl}formamido)propanoic acid
1-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)piperidin-4-amine
4-(4-cyclopropanecarbonyl-2-fluorophenyl)-3-methyl-1H-pyrazole
N-butyl-1-{1,3-dioxo-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
2-fluoro-N-(2-methoxyethyl)-N-propyl-5-sulfamoylbenzamide
N-methyl-2-(pyridin-2-yl)-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{4-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl}pyridine
N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)methyl]benzene-1-sulfonamide
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(pyridin-4-yl)acetamide
1-(1-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
1-cycloheptyl-N-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
N4-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
[(3-{[1-(2,6-dimethoxybenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-5-ylmethyl)amine
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
7-(cyclobutylmethyl)-2-methanesulfonyl-2,7-diazaspiro[4.5]decan-6-one
dimethyl({[1-methyl-2-(2-methylpropyl)-7-(3-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]sulfamoyl})amine
1-(2-phenylethyl)-3-(propan-2-yl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]ethyl}piperazine
N2,N2,5,6-tetramethyl-N4-(1-methylpiperidin-4-yl)pyrimidine-2,4-diamine
2-(2-methylpropyl)-8-(2-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[5-(6-methoxypyridin-3-yl)-1H-indol-1-yl]acetamide
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl][(5-methylthiophen-2-yl)methyl]amine
{2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)phenoxy]ethyl}dimethylamine
5-(methoxymethyl)-N-(4-{5-methyl-4-[(4,4,4-trifluorobutanamido)methyl]-1,3-oxazol-2-yl}phenyl)thiophene-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-[(4-ethoxyphenyl)methyl]cyclopropanamine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
3-{2-[(3-methoxyphenyl)methyl]morpholine-4-carbonyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1,2-oxazole-5-carboxamide
N,6,6-trimethyl-5-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]thiomorpholine-3-carboxamide
3-fluoro-4-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)benzamide
N3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-1,3-dicarboxamide
N3-[(1R)-1-(4-methoxyphenyl)ethyl]-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2-chlorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
3-(5-methylthiophen-2-yl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)-1H-pyrazole-5-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine-4-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(2-methoxyphenyl)methyl]piperazine
8-methoxy-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-{[3-(pyridin-2-yl)phenyl]methyl}morpholin-3-yl)acetic acid
3-{1-[1-(4-fluorophenyl)propan-2-yl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide