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(1R,5R)-N,N-dimethyl-6-[2-(2-methylphenoxy)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
5-(furan-2-ylmethyl)-5-{3-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methoxybenzoyl)piperidine
N-cyclopropyl-4-oxo-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-[(2,4-dimethoxyphenyl)methyl]-4-{4-[4-(pyridin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazol-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(1H-pyrazol-1-yl)acetamide
5-{4-[2-(benzyloxy)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
3-{[(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-N-ethylpyrimidin-2-amine
N-{[7-fluoro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(trifluoromethyl)benzamide
N-(furan-2-ylmethyl)-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(thiophen-2-ylmethyl)acetamide
(1S,4S)-5-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-[(4-benzylpiperidin-1-yl)methyl]-4-(3,6-dimethylpyrazin-2-yl)phenol
(2R)-2-[({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]-2-phenylethan-1-ol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(oxolan-3-ylmethyl)piperidine
7-[(4-fluorophenyl)methyl]-2-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenylpiperidin-4-ol
2-({ethyl[2-(morpholin-4-yl)ethyl]amino}methyl)-4-methylphenol
N-methyl-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(1,3-thiazol-2-yl)ethyl]propanamide
methyl (2S,4S)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-(furan-2-ylmethyl)-N-methylpyridin-2-amine
2-(3-methoxypropyl)-8-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(2-methoxyethyl)piperazine
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
4,5-dimethyl 1-[(3S,5S)-1-[(3,4-difluorophenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
(5S,9aS,9bS)-5-[2-(methylsulfanyl)pyrimidin-5-yl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3S,4S)-4-cyclopropyl-1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
N-cyclooctyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
4-[(2-fluorophenyl)methyl]-9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4S)-N-ethyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
N-cyclopropyl-5-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-2-methylpyrimidine
3-({[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
1-(cyclopropylmethyl)-5-[(4-hydroxyphenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl (2S)-1-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate
2-phenyl-1-[4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,3-thiadiazole-4-carboxamide
(1S,5R)-3-methyl-6-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}pyridine
3-(1-methyl-1H-imidazol-2-yl)-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidine
ethyl 1-benzyl-5-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2-phenylethyl)piperidine-4-carboxylate
(1S,5R)-3-(3-phenylpropyl)-6-(1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-4-(5-methyl-1,3-thiazole-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[3-({4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-2,4,6-trimethylphenyl]ethan-1-one
1-(pyrimidin-2-yl)-4-[2-(pyrrolidin-3-yl)benzoyl]-1,4-diazepane
1-[4-(2H-1,3-benzodioxole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2,2-diphenylethan-1-ol