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4-[2-(2H-indazol-2-yl)acetyl]-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
(3R,4R)-4-(azepan-1-yl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-ol
2-[1-(1-benzofuran-5-ylmethyl)pyrrolidin-2-yl]pyridine
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-3-methoxyphenol
N-[3-(4-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}piperidin-1-yl)phenyl]pyridine-3-carboxamide
N-(2-{1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-2-yl}ethyl)acetamide
2-(3,4-dichlorophenyl)-4-[(3,4-dimethoxypyridin-2-yl)methyl]morpholine
(2S,4S)-N-ethyl-1-(1-methylpiperidin-4-yl)-4-[2-(thiophen-2-yl)acetamido]pyrrolidine-2-carboxamide
(4aS,8aR)-6-(2,3-dihydro-1H-inden-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(4aR,7aS)-4-[(3-hydroxyphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-chloro-N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-[4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]phenol
N-[1-(4-chlorophenyl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine-2,4-diol
5-(2-fluorophenyl)-N-(1-methoxypropan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[3-(2-fluorophenoxy)azetidin-1-yl]-5-methylpyrimidine
4-methyl-1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidine-4-carboxylic acid
4-{[3-(5-methylfuran-2-yl)phenyl]methyl}thiomorpholine
2-[N-(3-fluorophenyl)methanesulfonamido]-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
(3S,4S)-3-({[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione
2-(butylsulfanyl)-6-[4-(morpholine-4-carbonyl)piperidin-1-yl]pyrimidin-4-amine
N-(2-methoxy-5-{[propyl(pyridin-3-ylmethyl)carbamoyl]amino}phenyl)acetamide
5-[(2-fluorophenyl)methyl]-5-(1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
4-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-5,6-dimethylpyrimidine
N-[2-(5-methylfuran-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
(4aS,7aR)-1-(4-methyl-1H-pyrrole-2-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-(4-chlorophenoxymethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
8-chloro-N-[(2,4-dihydroxyphenyl)methyl]-2-methylquinoline-4-carboxamide
N-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-N-(pyridin-4-ylmethyl)cyclopropanamine
6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(morpholin-4-yl)pyrimidin-4-amine
N-(1-ethyl-1H-indazol-3-yl)-2-[5-(1-phenylcyclopropyl)-2H-1,2,3,4-tetrazol-2-yl]acetamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclobutanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3-methoxyphenyl)methyl]-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-benzyl-1-methyl-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-{[4-(5-fluoro-2-methylphenyl)phenyl]sulfanyl}acetamide
14-(2-chloro-4-hydroxyphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
5-[4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)phenoxymethyl]furan-2-carboxylic acid
N-(3-hydroxypropyl)-1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
5-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-[(2R,3R)-2-hydroxy-1'-[(2-hydroxy-3-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
ethyl 5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
5-[({[3-(2-{4-[3-(2-methoxyphenyl)propanoyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
(1S,6R)-9-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one