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4-[({4-methyl-5-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-(cyclopropylmethyl)-8-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-2-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]pyridine-4-carboxamide
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3,3,3-trifluoro-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-(adamantan-1-ylmethyl)-N-(2-hydroxyethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
methyl 1-{2-hydroxy-3-[4-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
4-(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}piperidin-1-yl)-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
4-(3,5,7-trimethyl-1H-indole-2-amido)oxane-4-carboxylic acid
ethyl 3-[(2-fluorophenyl)methyl]-1-(quinoxaline-5-carbonyl)piperidine-3-carboxylate
2-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-1,3-thiazole-4-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[4-(benzyloxy)piperidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(1S,4S)-2-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-2-azabicyclo[2.2.1]heptane
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(1-methylpiperidin-4-yl)pyrimidin-2-amine
4-(2,6-dimethoxypyridine-3-carbonyl)-3,4-dihydro-2H-1,4-benzoxazine
N-[(5-fluoro-1H-indol-2-yl)methyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylformamido)-N-(2,5-dimethylphenyl)propanamide
2-methyl-4-(2-methylphenyl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-3-ol
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
3-chloro-4-(1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-1H-imidazol-2-yl)phenol
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
2-({[(3R,4R)-1-(3,5-difluoropyridine-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
7-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}quinolin-8-ol
1-[(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
N-(2-fluoro-4-methylphenyl)-2-{[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazol-4-yl]formamido}acetamide
5-{2-[6-(dimethylamino)pyridin-3-yl]-1H-imidazol-1-yl}-1,3,6-trimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-[1-(3-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}pyrimidin-2-amine
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
9-(cyclopropylmethyl)-4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(thian-4-yl)piperazine
1-[3-(1-methylpiperidin-3-yl)propanoyl]-4-phenylpiperidine-4-carboxylic acid
1-(2-methoxyethyl)-4-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}pyrrolidin-2-one
3-cyano-N-methyl-N-[3-(oxolan-2-yl)propyl]benzamide
ethyl 4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine-1-carboxylate
5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
3-(4-methyl-1,3-thiazol-5-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
methyl 2-{[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]sulfonyl}benzoate
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
5-[(4aS,8aR)-decahydroisoquinolin-2-yl]-1-[2-(benzenesulfonyl)ethyl]azepan-2-one
N-[(4-hydroxyazepan-4-yl)methyl]quinoline-6-carboxamide
2-methyl-N-(3-methylphenyl)-2,8-diazaspiro[4.5]decane-8-carboxamide
N-(2-methoxyethyl)-N-[(2-methoxyphenyl)methyl]-2-methyl-1,3-benzothiazole-6-carboxamide
(1R,2S,6R,7S)-4-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane