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3-{[4-(3-chlorophenyl)-5-{[methyl(quinolin-5-ylmethyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
3-(3-cyano-4-methylphenyl)-1-methyl-1-(thian-4-yl)urea
6-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
N-[(1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
ethyl 2-({4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carbonyl}amino)acetate
2-methyl-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}-1,4-diazepan-5-one
N-cycloheptyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(furan-2-yl)ethyl]piperidine-4-carboxamide
8-(1H-indol-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[6-hydroxy-4-(pyrazin-2-yl)-1,4-diazepane-1-carbonyl]-1H-pyrrole-3-carbonitrile
3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1H-pyrrole-2-carbonyl)piperidine
3-({1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
2-(4-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperazin-1-yl)ethan-1-ol
1-(azepan-1-yl)-3-[3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
8-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[1-tert-butyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-ethylpiperazin-2-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
4-[4-(azocane-1-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(2,6-difluorophenyl)methyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
8-(1,3-benzothiazol-2-ylmethyl)-3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R)-2-amino-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
5-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
(2S,4S)-4-amino-1-[(2-hydroxy-4-methylquinolin-6-yl)sulfonyl]-N-methylpyrrolidine-2-carboxamide
N-(1-benzofuran-2-ylmethyl)-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-cyclopropanecarbonyl-9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-[1-(2-phenylethyl)piperidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{4-[4-(4-methoxyphenyl)butan-2-yl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclopropyl-N-{2-phenyl-1-[1-(quinolin-6-ylmethyl)piperidin-4-yl]ethyl}furan-2-carboxamide
(5S,9aS,9bS)-5-[1-(4-methylphenyl)-1H-pyrazol-4-yl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 3-(3,4-dimethoxybenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-cyclopentyl-N-[2-(3-methylpiperidin-1-yl)ethyl]pyrimidin-2-amine
N-(2-hydroxy-2-phenylethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methylpiperidine-3-carboxamide
3-{1-[1-(cyclohexylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
N-(furan-2-ylmethyl)-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,4-dithiepan-6-amine
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(thiophen-3-yl)acetamide
6-methoxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]pyrimidin-4-amine
7-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
N,3-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-propyl-1-benzofuran-2-carboxamide
3-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-[(5-methylfuran-2-yl)methyl]-4-phenyl-1,4-diazepane
2-[4-(1H-pyrazole-4-carbonyl)piperazin-1-yl]pyrimidine
1-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-methylpiperazine
2-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
1-(3-chloro-4-methoxyphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
1-{4-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
1-[2-(4-phenylpiperidin-1-yl)ethyl]-3-(5-propyl-4H-1,2,4-triazol-3-yl)urea
N-cyclohexyl-2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
4-[(2-fluoro-4-methoxyphenyl)methyl]-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one