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2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[4-(pyrrolidin-1-ylmethyl)phenyl]-2-(pyrrolidin-3-yl)benzamide
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
5-{1-[5-(3-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
2-(4-methyl-3-phenyl-1H-pyrazol-1-yl)-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
5-methoxy-1-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-indole-2-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(cyclopropylmethyl)piperidine-4-carboxamide
N-{[1-(2-acetylbenzoyl)piperidin-3-yl]methyl}-2-chlorobenzamide
3-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-indole
2-[3-oxo-9-(pyrrolidine-1-carbonyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
1-(4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2-methylphenyl)-1H-pyrrole
N-[(1-cyclohexylpiperidin-3-yl)methyl]-5-phenyl-N-(pyridin-3-ylmethyl)pentanamide
N-({7-[2-(4-chlorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyrrolidine-1-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(cyclohexylmethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
(3R,4R)-1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
3-methyl-3-phenyl-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-3,5-dimethyl-1H-pyrazole
4-[(3-fluorophenyl)methyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(4-methoxyphenyl)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]furan-2-carboxamide
(1R,5R)-6-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
8-(2-methyl-1,3-thiazole-4-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-3-[1-(5-methyl-1,3,4-oxadiazole-2-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[1-(cyclohexylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
(3aS,6aS)-2-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-5-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-3-(4-chloro-2-fluorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl(pyridin-3-ylmethyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(3S,9aR)-3-[(benzyloxy)methyl]-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
4-{[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl](pyridin-3-yl)methyl}morpholine
N-({5-[(7-hydroxyquinolin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-[(3S)-1-[7-acetyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
5-(1H-indol-1-ylmethyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-1H-pyrazole-3-carboxamide
3-[(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-methylazepane-2-carboxamide
4-(benzyloxy)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
3-[(3-fluorophenyl)methyl]-N-methyl-N-[2-(oxan-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carbonitrile
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-(furan-3-ylmethyl)piperidine
1-[2-({[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one