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N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2,1,3-benzothiadiazole-4-sulfonamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylpropanamide
N3-(adamantan-1-yl)-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-[1-(2-hydroxybutyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4S)-N-ethyl-4-{[(3-methylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-({[1-(piperidin-1-yl)cyclohexyl]methyl}amino)-1λ4-thian-1-one
2-[(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetamide
2-(2-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}phenoxy)propanoic acid
6-{1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
3-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]benzoic acid
7-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-3-methyl-3,4-dihydroquinazolin-4-one
N,N-dimethyl-4-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]benzamide
5-phenyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(3-hydroxy-3-methylbutyl)benzamide
N-(4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}phenyl)acetamide
3-{[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}propane-1,2-diol
1-(4-{[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[4-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)thiophen-2-yl]ethan-1-one
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
3-(2-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenyl-N-(propan-2-yl)propanamide
N-[2-(diethylamino)ethyl]-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-6-(propan-2-yl)pyrimidin-2-amine
(2S)-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]-2-phenylbutanamide
(5R)-5-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}pyrrolidin-2-one
ethyl 1-(benzylcarbamoyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
4-methyl-14-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
ethyl 4-[4-(4-{[(4-fluorophenyl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
4-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}-N-methylbenzene-1-sulfonamide
(2R,3R)-3-{[(3-fluorophenyl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}morpholine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-methyl-5-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-2-(propan-2-yl)pyrimidine
2-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-3-methylquinoxaline
(5S,9aS,9bS)-5-(4-ethynylphenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
methyl 3-[(2,6-difluorophenyl)methyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
5-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-amino-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-6-methylpyrimidine-4-carboxamide
2-({4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(2-methylpropyl)-5-[(3,4,5-trimethoxyphenyl)methyl]-1H-1,2,4-triazole
2-(adamantan-1-yl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)acetamide
diethyl({[3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
N-[5-(1H-pyrazol-3-yl)quinolin-8-yl]acetamide
1-cyclohexyl-N-(1-propylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
4-methyl-7-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-1,2-dihydroquinolin-2-one
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]azocane