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{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-(cyclohex-3-ene-1-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
4-{[4-(furan-3-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzoic acid
methyl 2-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-3-(thiophen-3-yl)propanamide
1-(2-methyl-1,3-thiazole-4-carbonyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
(2S,4R)-4-amino-N-(furan-2-ylmethyl)-N-(2-phenylethyl)pyrrolidine-2-carboxamide
(3aR,6aR)-2-cyclopentyl-5-[(6-methoxypyridin-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[(5-methylfuran-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(3R,4R)-4-(morpholin-4-yl)-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-ol
N-methyl-2-(4-phenylpiperidin-1-yl)-N-(quinolin-5-ylmethyl)acetamide
4-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]pyrimidine-5-carboxylic acid
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-3-phenylprop-2-ynamide
1-(3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)-1H-pyrazole
(2S,4R)-N-ethyl-1-(naphthalen-2-ylmethyl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
6-({[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-2-methylpyrimidin-4-ol
8-(3-carbamoylpyridin-2-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl[(3-methylthiophen-2-yl)methyl][(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)spiro[2.2]pentane-1-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-ethyl-4-{[4-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N3-[furan-2-yl(phenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-chloro-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
ethyl 2-[methyl({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]acetate
1-({3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl}methyl)azepan-3-amine
N-[(3-fluorophenyl)methyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
4-[(4-methanesulfonylphenyl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-[1-butyl-5-(oxan-2-yl)-1H-1,2,4-triazol-3-yl]benzamide
3-(tert-butylsulfamoyl)-N-(3-fluorophenyl)-5-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}benzamide
1-[(6-ethoxyquinolin-2-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-(1-methanesulfonylpiperidin-4-yl)acetamide
2-(cyclopropylmethyl)-8-[2-(propan-2-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(1,4-oxazepane-4-carbonyl)-1-[4-(propan-2-yl)phenyl]pyrrolidin-2-one
N-methyl-N-(piperidin-3-ylmethyl)-3-[(thiophen-2-ylmethyl)amino]benzamide
(1S,4S)-2-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-2-azabicyclo[2.2.1]heptane
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
2-(1-benzothiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
methyl (2S)-1-{2-[4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]pyridine
N-[2-(cyclohexylsulfanyl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]-6-phenyl-2,3-dihydropyridazin-3-one
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-{[(4-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-(1H-1,3-benzodiazol-2-yl)-2-({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}amino)acetamide
N-[(1R,2S)-2-phenylcyclopropyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
4-{4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]piperazin-1-yl}-6-methylpyrimidin-2-amine
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-(2-methoxyethyl)-4-{[(3-methoxyphenyl)methyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine