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N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-ethoxyacetyl)pyrrolidin-3-yl]pyridine-3-carboxamide
3-(cyclopropylmethyl)-1-(thiophen-3-ylmethyl)piperidine-3-carboxylic acid
8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-butyl-4-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
1-{9-[(2-methoxy-4-methylphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl}-2-methylpropan-1-one
N-(2-methoxyethyl)-1-{1-[(4-methoxypyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
(benzylsulfamoyl)(2,3-dihydro-1-benzofuran-2-ylmethyl)methylamine
2-amino-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
1-[3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzenesulfonyl]azepane
N,1-dimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-4-oxo-1,4-dihydroquinoline-3-carboxamide
(1S,4S)-2-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-2-azabicyclo[2.2.1]heptane
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(1-methylpiperidin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3,6-dimethyl-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
[(2,5-dimethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-{2-[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4-methylpyridin-2-amine
[(3R,4R)-1-{5-[(dimethylamino)methyl]furan-2-carbonyl}-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
3-[1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2-ethyl-1,3-dihydroxypropan-2-yl)acetamide
1-[(2-fluorophenyl)methoxy]-8-(2,7,8-trimethylquinoline-4-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
4,6-dimethyl-2-({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}amino)pyridine-3-carbonitrile
1-[5-(methoxymethyl)furan-2-carbonyl]-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
3-{[2-(5-propylfuran-2-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
methyl 5-oxo-5-[(2R,3R)-3-propanamido-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]pentanoate
2-methyl-4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
[3-(1H-1,2,3-benzotriazol-1-yl)propyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-(7-methoxy-4-methylquinazolin-2-yl)-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
N-methyl-6-oxo-4-[2-(propan-2-yl)-1,3-oxazol-4-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(2-methylpyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-butyl-N-methylacetamide
{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}urea
8-[(3,4-dimethoxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]phenyl}but-3-yn-1-ol
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]cyclohex-3-ene-1-carboxamide
{1-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
1-(3-methylphenyl)-3-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]urea
3-(3-methoxyphenyl)-3-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(3-phenylpropyl)acetamide
N-[(3-fluorophenyl)methyl]-2-(1H-imidazol-4-yl)-N-[(4-methoxyphenyl)methyl]acetamide
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)furan-3-carboxamide
1-ethyl-4-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrazole
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-phenylpiperazine
N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(1,3-dihydro-2-benzofuran-5-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-3-ylmethyl)urea
1-cyclopropyl-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
methyl 4-methyl-3-({[3-(1H-1,2,3-triazol-1-yl)propyl]carbamoyl}amino)benzoate