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methyl 8-({4-[methyl(phenyl)amino]phenyl}methyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(3-hydroxyphenyl)-1-{3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}propan-1-one
4-benzyl-3-ethyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,4-diazepan-5-one
1-(5-acetyl-2-methoxyphenyl)-3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
3-{5-[(1-methyl-1H-1,2,3-benzotriazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
5,6-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-cyclopentyl-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}acetamide
ethyl 1-benzyl-5-[(3,4-difluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(4-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
4-fluoro-N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(4-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}quinazolin-2-yl)ethan-1-amine
N-(2-methoxy-2-methylpropyl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-3-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanamide
4-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)benzonitrile
2-{4-[(2-chloro-4-fluorophenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-(benzyloxy)-8-[2-(2-chlorophenoxy)acetyl]-1,8-diazaspiro[4.5]decan-2-one
(4aS,7aR)-1-(2,3-dimethylbenzoyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(3S)-3-benzyl-4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperazin-2-one
N-[1-(7-{[5-(hydroxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]pyridine-2-carboxamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
3-(but-2-yn-1-yl)-5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
2-amino-6-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
2-ethyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyrimidine-5-carboxamide
2-(1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}pyrrolidin-2-yl)ethan-1-ol
N-benzyl-N-methyl-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}propanamide
N-(3-hydroxypropyl)-1-[1-(naphthalen-1-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-ethyl-2-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyrimidin-4-amine
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-[1-(3-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
1-(1-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)-4-methylpiperazine
N-[2-(2,4-difluorophenyl)-1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]propanamide
3-[(3R,4S)-1-[2-(4-methylphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-4-carbonitrile
4-[2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-ethyl-3-(4-phenyl-1-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-imidazol-5-yl)piperidine
4-(azepane-1-carbonyl)-6-chloro-2-(1H-pyrazol-4-yl)quinoline
1-[3-(furan-2-yl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
2,7-dimethyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-(cyclopropylmethoxy)-4-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N,N-dimethyl-2-({3-[(oxolan-3-ylmethyl)sulfamoyl]phenyl}formamido)acetamide
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-(methoxymethyl)thiophene-2-carboxamide
5-[methyl(2-phenylethyl)amino]-2-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,3-dihydropyridazin-3-one
N-[2-(3-chlorophenyl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2,5-dimethyl-N-({7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-3-carboxamide
9-[(2,5-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-ethoxy-4-methyl-2-{2-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrrolidin-1-yl}quinazoline
2-amino-3-ethyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-chloro-N-[1-(2,5-difluorophenyl)cyclopropyl]-3-methyl-1H-pyrazole-5-carboxamide