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6-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N,N-diethyl-1-{3-[(3-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}piperidine-3-carboxamide
3-methyl-5-(phenoxymethyl)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]furan-2-carboxamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(pyrrolidine-1-carbonyl)piperidine
N-methyl-3-(pyridin-3-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
2-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1,3-benzothiazole-5-carboxamide
N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N-benzyl-2-[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
1-[2-({[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-3-ol
N-(2-methoxyethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(propan-2-yl)acetamide
1,3-dimethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-methyl-1-[(5-methyl-1H-imidazol-4-yl)methyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
(3R,5R)-N-[3-(4-chlorophenyl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[4-(cyclopropylmethyl)piperazin-1-yl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
1-(4-{[(1-methylpiperidin-4-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
8-(6-cyclopropylpyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]carbamoyl}methyl)-1,2,3-oxadiazol-3-ium-5-olate
2,6-difluoro-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-methyl-6-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
4-hydroxy-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
8-(2,7,8-trimethylquinoline-4-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-{[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
3-hydroxy-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-2-carboxamide
8-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-2-carboxamide
methyl 1-{9-methoxy-3-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
methyl (2S)-4-methyl-2-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamido}pentanoate
N-[4-(2H-1,3-benzodioxol-4-yl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methoxyacetamide
4-(dimethyl-1,2-oxazole-4-carbonyl)-2-(naphthalen-1-ylmethyl)morpholine
(2R)-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyloxolane-2-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-(cyclohexylmethyl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[3-(2-ethylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{4-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-3-carboxamide
4-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperazin-2-one
4-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}benzonitrile
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(carbamoylmethyl)piperidine-4-carboxamide
2-[({1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
(4aR,8aR)-2-(2-aminopyridine-4-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
3-[(1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)methyl]benzoic acid
N-methyl-N-{1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-2-phenylethyl}thiophene-2-carboxamide
3-[1-(2-ethylpyridine-4-carbonyl)piperidin-3-yl]benzoic acid
3-methyl-2-{1-[4-(3-methyl-1-benzofuran-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}pyridine
5-benzyl-5-(1-cyclobutanecarbonylpiperidin-4-yl)-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-N-[1-(pyrimidin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(3-cyanophenyl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(2-{7-[(2-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-3-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]amine
3-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-5,6-dimethyl-1,2-dihydropyridin-2-one