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(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(4-methyl-3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(2-chlorophenyl)-3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-(2-fluorophenyl)-4-[(3-{[1-(pyridine-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
(2E)-N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(furan-2-yl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}prop-2-enamide
5-methyl-14-[2-(prop-2-en-1-yloxy)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
methyl 4-({3-[2-(furan-2-ylformamido)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)benzoate
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-2-phenylpyrrolidine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H-indole-6-carboxamide
1-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-4-phenylpiperazine
3-acetamido-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]propanamide
2-{5-[(benzyloxy)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
2,4-dichloro-3-{[3-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}phenol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylpyrimidin-4-amine
5-butyl-1'-[4-(trifluoromethyl)pyridin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}pyridine-2-carbonitrile
3-[(3-methoxyphenyl)methyl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-N-methyl-N-[2-(methylamino)ethyl]benzene-1-sulfonamide
1'-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methanesulfonylpyrrolidine-2-carboxamide
4-(4-fluoro-3-methylbenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
8-[(3-fluorophenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-benzyl-8-[(2,2-dimethyloxan-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
[(3-methoxyphenyl)methyl]({[5-(oxolan-2-yl)thiophen-2-yl]methyl})(prop-2-en-1-yl)amine
(1R,5R)-6-(2-methoxyethyl)-3-[3-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-(5-propyl-1,3,4-thiadiazol-2-yl)-2-({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}amino)acetamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
3-chloro-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-{[(2E)-2-methylbut-2-en-1-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
2-(4-fluoro-2-methoxyphenyl)-2-(4-methyl-1,4-diazepan-1-yl)acetic acid
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)methylamine
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
N-[(2R,3R)-1'-(3-chlorothiophene-2-carbonyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-methyl-3-[methyl({[6-(trifluoromethyl)pyridin-3-yl]methyl})amino]butanamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
3-chloro-6-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}pyridine-2-carboxylic acid
1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-6-ol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(4-fluorophenyl)methyl]-N-propylacetamide
2-[5-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-3-yl]phenol
N,N-diethyl-3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-[3-(propan-2-yloxy)propyl]pyrrolidin-2-one
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
9-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(4-{4-[(2-acetamidoethyl)amino]piperidin-1-yl}phenyl)-4-methoxybenzamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-3-yl]propan-1-ol
4-[5-({ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
N-[(2-chloro-6-fluorophenyl)methyl]-2-propyl-1,3-thiazole-4-carboxamide