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4-{1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]azetidin-3-yl}pyridine
3-(2H-1,3-benzodioxol-5-yl)-N-[(1-hydroxycyclohexyl)methyl]-3-phenylpropanamide
1-(morpholin-4-yl)-3-[1-(quinoline-6-carbonyl)piperidin-4-yl]propan-1-one
N-(4-{4-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl})amine
3-[({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}oxy)methyl]pyridine
N-ethyl-4-oxo-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}adamantane-1-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}acetamide
(1S,5R)-3-(3-phenylpropyl)-6-(trimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(benzyloxy)azetidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
(2S,4R)-4-(dimethylamino)-1-[3-(2,2-dimethylpropanamido)-4-methylbenzoyl]pyrrolidine-2-carboxylic acid
2-(2,3-dihydro-1-benzofuran-7-yl)-2-({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)acetic acid
2-hydroxy-4-methoxy-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)benzamide
1-(2-methoxyethyl)-8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-ol
3-phenyl-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
N-[2-(2,3-dimethoxyphenyl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
(2H-1,3-benzodioxol-4-ylmethyl)(ethyl)[2-(morpholin-4-yl)ethyl]amine
1-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-ol
3-(2-amino-4-methyl-6-{[(3-methylphenyl)methyl]amino}pyrimidin-5-yl)propanoic acid
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}amine
3-(2-hydroxypyridin-3-yl)-1-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]urea
(4aS,7aR)-1-[(6-methylpyridin-2-yl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-amino-3-ethyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2,4-dichloro-6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenol
2-{1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylacetamide
N-[(2,6-difluorophenyl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(morpholine-4-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-N-[1-(2-fluorophenyl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
2-{1-[(4-methylphenyl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
1-(2-chloro-6-methylphenyl)-3-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
8-cyclopropanecarbonyl-2-[(2-fluoro-5-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 8-[(2,4-dimethoxyphenyl)methyl]-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
11-{[(2-benzyl-1,3-thiazol-4-yl)methyl]amino}-4-(3-methylbutyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(pyridin-2-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidin-2-amine
2-[(4-ethoxyphenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[3-(cycloheptylamino)butyl]phenol
3-[3-(dimethylamino)propyl]-8-(oxolan-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(2-ethylbutyl)({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-methoxypropanamide
2-(2-methoxyphenyl)-N-[4-(pyridin-3-yloxy)phenyl]acetamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(3-phenylpropyl)piperidine
3-ethyl-3-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[2-(1H-pyrazol-1-yl)phenyl]urea