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N-[1-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
{3-[(4-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}methanol
2-(dimethylamino)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(2,2-dimethylpropanoyl)piperidine-3-carboxylate
[2-(2,6-dimethylphenoxy)ethyl](ethyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
2-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-6-methylpyridine
2-(2-chloro-4-fluorophenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
1-ethyl-4-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}-1H-pyrrole-2-carbonitrile
2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}pyrazine
8-[2-(4-chlorophenoxy)acetyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
1-(furan-2-ylmethyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-(4-fluorophenyl)-4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperazin-2-one
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]isoquinoline
6-methyl-4-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}-1,2-dihydropyridin-2-one
2-[4-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
(2S,4R)-1-(adamantan-2-yl)-4-[(4-methoxyphenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(2,3-difluorophenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-butyl-3-methyl-5-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
N-(2-oxoazepan-3-yl)-3-(1H-pyrazol-4-yl)benzamide
5-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
3-methyl-1-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}butan-1-ol
2-cyclopentyl-2-phenyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
5-methyl-N-[2-(methylsulfamoyl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
6-ethyl-2-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-4-carboxamide
(3aR,5R,6S,7aS)-2-(2-hydroxynaphthalene-1-carbonyl)-octahydro-1H-isoindole-5,6-diol
6-(2-cyclopropylacetyl)-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(3-fluorophenyl)ethyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-9H-purine
4-fluoro-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
8-(1-ethyl-6-oxopiperidine-3-carbonyl)-2-(3-methylbutyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-[3-(dimethylamino)propyl]piperidine-3-carboxamide
N-({3-methyl-7-[3-(3-methylphenyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
N-[1-({[(1-benzyl-1H-pyrazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-4-oxo-4-phenylbutanamide
5-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
(1r,4r)-4-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]cyclohexan-1-ol
N-(2,3-dihydro-1H-inden-4-yl)-4-{[3-(hydroxymethyl)morpholin-4-yl]methyl}benzamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(4-methoxyphenyl)furan-2-carboxamide
1-benzyl-8-[(4-ethylphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetamide
5-ethyl-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclopentanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-phenoxypropan-1-one
N-[(3-chlorophenyl)methyl]-1-[(2,6-difluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid