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3-{2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-methyl-N-(propan-2-yl)-2-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[(3-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
1-[4-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-methyl-N-(2-methylpropyl)-3-(naphthalen-1-ylmethyl)-1,2-oxazole-5-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohex-1-ene-1-carboxamide
N-(1-benzylpiperidin-4-yl)-5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-amine
1-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
3-(2-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-benzyl-5-[(2-fluorophenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(carbamoylmethyl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxamide
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(2-methylphenyl)methyl](prop-2-en-1-yl)amine
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-3-cyclopropylpropanamide
5-ethyl-N4-[1-(pyridin-3-yl)propyl]pyrimidine-2,4-diamine
3-[2,4-dichloro-3-(pyrrolidin-1-ylmethyl)phenoxy]-2,5-dimethylpyrazine
3-hydroxy-1-(2-methoxyethyl)-3-{[methyl(quinolin-6-ylmethyl)amino]methyl}piperidin-2-one
4-ethyl-2-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-thiazole-5-carboxamide
1-[4-({3-[4-(1-hydroxypropyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
methyl 3-[(3,5-difluorophenyl)methyl]-9-[3-(dimethylamino)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-hydroxy-3-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[1-(pyridin-4-yl)propyl]propanamide
8-fluoro-2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]quinoline
N-[(3-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-2-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
N-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
4-amino-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-hydroxybutan-1-one
1-[4-(piperidin-1-ylmethyl)piperidin-1-yl]-3-(1H-pyrrol-1-yl)propan-1-one
1-{4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]thiophen-2-yl}ethan-1-one
1-(7-fluoro-1,2,3,4-tetrahydroisoquinolin-2-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
ethyl 4-[(4-chlorophenyl)methyl]-1-(1-ethylpiperidine-3-carbonyl)piperidine-4-carboxylate
3-({[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
6-methoxy-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrimidin-4-amine
1-methyl-5-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(2-methoxyethyl)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-cyclohexanecarbonyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
7-cyclopentyl-2-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[3-(1H-imidazol-1-yl)propyl]-9-(1-methyl-1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
8-methyl-3-(3-phenylpiperidine-1-carbonyl)-4H-pyrido[1,2-a]pyrimidin-4-one
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(propan-2-yl)amine
5-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-[(3S,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
N-(1-{1-[2-(3-chlorophenoxy)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
2,7-dimethyl-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(4-cyclopropanecarbonylphenyl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[(1E)-pent-1-en-1-yl]-1-phenyl-1H-1,2,3,4-tetrazole
N-{3-[6-amino-5-cyano-4-(3-ethenylphenyl)pyridin-2-yl]phenyl}acetamide