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5-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-fluoro-4-{[4-(2-fluorophenoxy)piperidin-1-yl]methyl}-6-methoxyphenol
5-(2,4-difluorophenoxymethyl)-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
(2S,4R)-4-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
ethyl 4-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}amine
methyl 2-{[(2-chlorophenyl)methyl]sulfamoyl}-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-cyclopropanecarbonyl-1'-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(1H-pyrazol-3-yl)piperidine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]cyclohexanecarboxamide
2-(6-hydroxyhexyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
methyl 2-oxo-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxoethyl}acetamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2,5-dihydro-1H-pyrrole-2-carboxamide
N-(1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
(2R,3R,6R)-3-(4-methylphenyl)-5-[(2-propylpyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2,5-dimethylphenyl)methyl]-3-methylpiperidine
3-(3,4-dimethoxybenzoyl)-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-3-ol
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1-methylcyclopropyl)acetamide
9-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[1-(thiophen-3-yl)propan-2-yl]pyrimidin-2-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperazine
3-(3-hydroxypropyl)-4-(2-phenylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(3-methoxyphenyl)propanamide
{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
4-methyl-5-{[1-(3-methylpyridin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-thiazol-2-amine
N-[(3-hydroxyphenyl)methyl]-N,3,5-trimethyl-1-benzofuran-2-carboxamide
N-[(3-fluorophenyl)methyl]-9-methoxy-3-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[2-(pyridin-2-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-6-fluoro-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-(4-{1-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
4-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3-methyl-1H-pyrazole-4-carboxamide
4-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}phenol
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
3-(2-amino-1,3-thiazol-4-yl)-1-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
3-(2-methoxybenzoyl)-1-[4-(trifluoromethyl)benzoyl]piperidine
(1-{4-[4-({[2-fluoro-5-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-yl)methanol
N-[(3,4-difluorophenyl)methyl]-2-methyl-4-phenylpyrimidine-5-carboxamide
4-hydroxy-3-methyl-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
2-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-9-oxa-2-azaspiro[5.5]undecane
N-{[4-(cyclooctyloxy)phenyl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(pyridin-3-ylmethyl)acetamide
N-(3-phenylpropyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(3-methylbutyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-chloro-N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
N-methyl-3-phenoxy-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
3-({[6,7-dimethoxy-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}(2-hydroxyethyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione