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4-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]-1,4-oxazepane
N-cyclopropyl-3-{1-[4-(propan-2-yloxy)benzoyl]piperidin-4-yl}propanamide
methyl 3-(4-ethenylbenzoyl)-9-[2-(morpholin-4-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(2-ethylbutyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-methyl-2-{5-methyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
1-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]azepan-2-one
4-methyl-2-oxo-5-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
4-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
3-amino-1-[3-(dimethylamino)-2,2-dimethylpropyl]pyrrolidine-3-carboxylic acid
9-[(4-acetylphenyl)methyl]-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[4-(2,3-dihydro-1H-isoindol-2-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[({[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)methyl]-1,3-thiazol-2-amine
1-(2-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)azepan-2-one
1-ethyl-5-({[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[5-(quinolin-8-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
2-(dimethylamino)-4-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrimidine-5-carboxamide
1-(2,6-dimethylpyridin-4-yl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
3-{5-ethyl-6-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}azepan-2-one
N-(dimethyl-1H-1,2,4-triazol-3-yl)-2-(4-methoxyphenyl)morpholine-4-carboxamide
(cyclohexylmethyl)({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
N-methyl-N-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)methanesulfonamide
1-(2,3-dimethyl-1H-indole-7-carbonyl)-N-phenylpiperidin-3-amine
3-[3-({[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
methyl 3-(2-acetylbenzoyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{2-[4-(3-methylbut-2-en-1-yl)morpholin-2-yl]ethyl}cyclopropanesulfonamide
N-[2-(2-chlorophenyl)-1-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
N-[2-(5-methyl-4-{[methyl(6-methylhept-5-en-2-yl)amino]methyl}-1,3-oxazol-2-yl)phenyl]methanesulfonamide
1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}-4-methyl-1,4-diazepane
N-[(2R,4R,6S)-2-cyclohexyl-6-[1-(2-methoxyethyl)-1H-imidazol-2-yl]oxan-4-yl]acetamide
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
1-benzoyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]piperidin-4-amine
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
N-[2-(3-ethylpiperazine-1-carbonyl)phenyl]-N-methylthiophene-2-carboxamide
3-methoxy-N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
methyl 7-oxo-9-[2-(thiophen-2-yl)ethoxy]-3-(4,4,4-trifluorobutanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S,4R)-4-amino-1-(3,5-dimethylbenzenesulfonyl)-N-ethylpyrrolidine-2-carboxamide
N-[(3S,4R)-1-[2-(2,4-dimethoxyphenyl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
(4aR,7aS)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(2-ethoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-chlorophenyl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-tert-butyl-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-[(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)oxy]pyridine
2-(4-ethoxyphenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[(2R,3R)-1'-(adamantan-2-yl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
2,3,5-trimethyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine