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N-cyclopentyl-1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(thiophen-2-yl)acetamide
N-(2-hydroxyethyl)-N-methyl-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
6-(1-ethylpiperidine-2-carbonyl)-3-(4-fluoro-3-methylphenyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
5-(3-acetylphenoxymethyl)-N-[(4-fluorophenyl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]propanamide
(2R)-2-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-(4-{[(2,2-dimethyloxan-4-yl)(ethyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
3-[1-(5-acetylthiophene-2-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
2-ethyl-4-(2-methylpyridin-4-yl)-1-(propan-2-yl)piperazine
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(2,3,4-trifluorophenyl)methyl]benzamide
1-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]pentane-1,4-dione
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(pyridin-3-ylmethyl)acetamide
6-hydroxy-4-[(3-methylquinoxalin-2-yl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3,5-dichloro-N-(1-methoxybutan-2-yl)-4-(prop-2-en-1-yloxy)benzamide
N-phenyl-1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)piperidin-3-amine
5-ethyl-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
8-cyclopentyl-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[5-(2-ethylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
2-(4-fluorophenyl)-N-[3-(pyrrolidin-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[3-(furan-2-yl)benzoyl]-N-[4-(1H-pyrazol-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-chloro-N-{[1-(1H-indole-5-carbonyl)piperidin-3-yl]methyl}benzamide
2-(4-chlorophenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
methyl 2-{[2-(cyclooctylcarbamoyl)ethyl]amino}-3-hydroxypropanoate
N-ethyl-1-{3-[ethyl(methyl)carbamoyl]benzenesulfonyl}pyrrolidine-3-carboxamide
2-{5-[2-(ethylamino)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}acetic acid
1-(2-cyclohexylethyl)-3-{[(furan-2-ylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
N-(1-{7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3,5-dimethylbenzamide
2-methyl-2-(thiophen-2-ylformamido)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
4-[(4-fluorophenyl)methyl]-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
[3-(cyclopropylmethyl)-1-[1-(morpholin-4-yl)cyclohexanecarbonyl]piperidin-3-yl]methanol
2-{2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-3-methylpyridine
4-ethyl-3-({1-[4-(ethylamino)pyrimidin-2-yl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-methylphenyl)-4-{spiro[2.5]octane-1-carbonyl}piperazin-2-one
(3S,4R)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
N-methyl-N-(2-phenoxyethyl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
methyl 4-oxo-4-(7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)butanoate
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[2-(pyridin-4-yl)ethyl]acetamide
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl)ethan-1-ol
3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-1-one
3-(4-{[(3S,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)prop-2-yn-1-ol
(2S,4S)-4-[4-({[(3-chloro-4-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide