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3-[1-(3-chloro-2-methylphenyl)-1H-imidazol-2-yl]-1-ethylpiperidine
N-[1-(furan-2-carbonyl)piperidin-4-yl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-[3-(2-phenylethyl)-1H-1,2,4-triazole-5-carbonyl]-1,2,3,4-tetrahydroquinoline
2-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-7-(4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}piperidin-4-amine
methyl (2R,4S)-1-(1,5-dimethyl-1H-indazole-3-carbonyl)-4-hydroxypiperidine-2-carboxylate
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[3-(2-methylpropoxy)phenyl]methyl}pyrrolidin-3-yl]methanol
3-(3-methoxyphenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]propan-1-one
4-({2-[1-(4-fluoro-3-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}urea
N-[2-(4-methoxyphenyl)ethyl]-3-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methylpiperidin-4-yl)methyl]propanamide
4-methoxy-N-[2-({4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}amino)ethyl]benzene-1-sulfonamide
1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-[2-(methylsulfanyl)benzoyl]piperidine
N-ethyl-2-methoxy-N-[2-(3-methylphenoxy)ethyl]butanamide
4-{1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
5-(methoxymethyl)-N-[(3-methoxyphenyl)methyl]-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
2-{5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}pyridine
2-ethyl-8-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(5-methylthiophen-2-yl)-1H-imidazole
5-[({[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
N-[(1-cycloheptylpiperidin-3-yl)methyl]-4-methoxybenzene-1-sulfonamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(furan-2-ylmethyl)piperidine-3-carboxamide
(1S,9S)-11-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-(1,3-dihydro-2-benzofuran-5-yl)-3-(2,5-dimethoxyphenyl)pyrrolidine-1-carboxamide
4-(2-aminopyrimidin-4-yl)-7-(1,3-benzothiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl[(2-fluoro-5-methoxyphenyl)methyl][(1-methyl-1H-imidazol-2-yl)methyl]amine
3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]benzonitrile
2-(1-ethylpiperidin-4-yl)-N-[1-(1,3-thiazol-2-yl)propyl]acetamide
N-(1,4-dioxan-2-ylmethyl)-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
6-(1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidin-3-yl)pyrimidin-4-ol
5-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)pyrimidine
1-(2-oxo-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
2-(2-methoxyphenyl)-5-(quinolin-6-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
N-cyclopentyl-2-ethyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}butanamide
N-(1,4-dioxan-2-ylmethyl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4-{[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]sulfonyl}-N-methylthiophene-2-carboxamide
8-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5,5-dimethyl-3-{2-oxo-2-[3-(1H-pyrazol-3-yl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
2-{[5-(1H-pyrazol-5-yl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-{1-methyl-4-[3-(piperidin-1-yl)azetidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
1-{[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]methyl}-3-ethylurea
N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[(2-methylphenyl)methyl]piperazine
cyclohexyl({4-[2-(methylsulfanyl)pyridine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
N-[2-(4-fluorophenyl)ethyl]-3-methyl-1-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
[(5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]dimethylamine
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
2-methyl-5-propyl-4-[3-(pyridin-2-yl)azetidin-1-yl]pyrimidine