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1-(4-butylphenyl)-3-[(5-methyl-1H-pyrazol-3-yl)methyl]urea
methyl 4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-methylpiperazine-2-carboxylate
5-(azepan-1-yl)-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4aR,8aS)-6-(2-phenoxyacetyl)-decahydro-1,6-naphthyridin-1-yl]-4,4,4-trifluorobutan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2-oxazole-5-carboxamide
3-fluoro-2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine
8-(5-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[3-(6-aminopyridin-3-yl)-1-(2-ethoxyphenyl)prop-2-yn-1-yl]piperidine-4-carboxamide
1-(2,4-difluoro-3-methoxybenzoyl)-4-[(3-methylphenyl)methyl]piperazine
3-(4-methyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-[2-(8-fluoroquinolin-2-yl)-1H-imidazol-1-yl]-3-(furan-2-yl)propanoic acid
5,7-dimethyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
(2S,4R)-1-(2,2-diphenylethyl)-4-{[(3-methoxyphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
6-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-{2-[(3-fluorophenyl)methyl]morpholine-4-carbonyl}quinoline
1-[(2-methoxynaphthalen-1-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-9H-purin-6-amine
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[3-(propan-2-yloxy)propyl]piperidine-3-carboxamide
1-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)carbamoyl}methyl)piperidine-4-carboxamide
(1R,2R,4R)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(piperidine-1-carbonyl)pyridine
(1R,2R,6S,7S)-4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-azatricyclo[5.2.1.02,6]decane
3,4,7-trimethyl-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
6-(cyclopropylamino)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-{2-[({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]ethyl}piperidin-4-ol
6-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1,3-thiazol-2-yl)piperidine
5-(3-fluorophenoxymethyl)-N-(1-methoxybutan-2-yl)-1H-pyrazole-3-carboxamide
1-({5-[(2-fluoro-4-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N,2,4-trimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1,3-oxazole-5-carboxamide
2-[5-methyl-4-(3-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
2-(2-fluoro-3-methylphenyl)-2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]acetic acid
N-benzyl-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}-N-methylpyrrolidine-3-carboxamide
9-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-ethoxy-6-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenol
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(1-benzyl-1H-imidazol-2-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
1-[(2,4-dimethylphenyl)methyl]-4-{furo[3,2-c]pyridin-4-yl}piperazine
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-cyclohexylurea
5-[5-(6-fluoroquinolin-2-yl)-4-phenyl-1H-imidazol-1-yl]pentan-1-amine
4-(3-propoxypiperidine-1-carbonyl)benzene-1-sulfonamide