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N-[3-(3-methoxyphenyl)phenyl]-1-(pentan-3-yl)piperidine-4-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-4-(4-methylpiperazine-1-carbonyl)pyridin-2-amine
1-(2-methyl-1H-pyrrole-3-carbonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-chloro-N-(2-hydroxyethyl)-1,5-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-3-carboxamide
4-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}benzonitrile
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-[(4-fluorophenyl)methyl]-4-[(2-methoxypyrimidin-5-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
(4aR,7aS)-1-(1H-imidazol-2-ylmethyl)-4-(4,4,4-trifluorobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-benzyl-4-(1H-1,2,3-triazole-5-carbonyl)piperazin-2-one
9-[2-(4-fluorophenyl)-2-hydroxyacetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl({[(2R,5S)-5-[(6-methoxypyridin-3-yl)methyl]oxolan-2-yl]methyl})[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-(ethylamino)-N-[2-(thiophen-2-yl)ethyl]pyrimidine-5-carboxamide
2-[1-(1-benzothiophene-2-carbonyl)-1,4-diazepan-6-yl]acetic acid
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
3-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-(2,3-dimethylquinoxalin-6-yl)urea
3-(1-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)-1,3-oxazolidin-2-one
3-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
6-(2-{1-butyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-2,3-dihydropyridazin-3-one
4-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
N-methyl-5-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
4-[4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propan-2-yl}acetamide
8-[(4-chlorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-(morpholin-2-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(1R,5R)-6-[(2,4-dichlorophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{2-[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amino]pyrimidin-4-yl}pyrrolidin-3-ol
1-[5-(4-chloro-1-methyl-1H-pyrrol-2-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
4-methyl-7-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazine
8-hydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}quinoline-7-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-acetamidopropanamide
N-methyl-N-(2-phenyl-1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}ethyl)thiophene-3-carboxamide
8-(2-hydroxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{2-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
11-{[(1-phenylcyclopentyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[4-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
5-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
2-({2-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]phenyl}amino)acetic acid
N-(2-methoxyethyl)-1-(3-methylbutyl)-5-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-[3-(furan-2-yl)propyl]-4-phenyl-1H-imidazole
[2-(2,4-difluorophenyl)ethyl](ethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3R,4S)-3,4-dimethyl-1-{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}piperidin-4-ol
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-[({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]benzene-1-sulfonamide
3-{2-oxo-2-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}imidazolidine-2,4-dione
3-(4-chlorophenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid