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3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
4-{1-[(5-ethylfuran-2-yl)methyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N'-cyclopentyl-N-(3-propoxypropyl)butanediamide
2-{[(2-fluorophenyl)methyl](methyl)amino}-N-(4H-1,2,4-triazol-4-yl)acetamide
1-(2,2-difluoroethyl)-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-5-(1H-indol-1-ylmethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
N,N-dimethyl-2-{[3-(pyridin-3-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl)amino}-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]acetamide
5-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,3-oxazole-4-carboxamide
3-({2-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-[3-(2-fluorophenyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-ethyl-4,6-dimethyl-3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
2,8-dimethyl-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}quinoline-4-carboxamide
1-(4-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}piperidin-1-yl)butan-1-one
{3-[(4-methyl-1H-imidazol-2-yl)methyl]-9-[3-(methylsulfanyl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
4-chloro-2-[(1E)-2-({3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}methyl)prop-1-en-1-yl]phenol
2-[(4-chlorophenyl)methyl]-8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
2-(2-fluorophenyl)-1-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-imidazole
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
5-(2-methoxyphenoxymethyl)-3-(2-methylpyrrolidine-1-carbonyl)-1H-pyrazole
1-[2-({[(3-fluorophenyl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
4-(2-methyl-1-benzofuran-5-carbonyl)-1λ6-thiomorpholine-1,1-dione
(1H-indol-7-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})methylamine
3-methoxy-1-(4-{4-[3-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)propan-1-one
1-[9-hydroxy-7-(thianthren-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
[(2S,6S)-4-(1,4-dithiepan-6-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
methyl 3-ethyl-2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3H-imidazo[4,5-b]pyridine-6-carboxylate
2-{3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
4-methyl-2-phenyl-1-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2,4-dimethoxybenzene-1-sulfonamide
9-(2,3-dihydro-1H-inden-2-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]acetamide
6-ethyl-N,1-dimethyl-N-[3-(oxolan-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-cyclobutyl-4-(furan-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
6-(2,5-dimethylfuran-3-yl)-N-(3-hydroxy-2,2-dimethylpropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6,7-dimethoxy-1-methyl-2-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
(2S,4R)-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-N-cycloheptyl-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-5-cyclopropyl-1,3-oxazole
3-(butan-2-yl)-1-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
N-(3-methoxypropyl)-6-[2-(pyridin-3-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[1-(2-methoxyethyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(4aS,8aS)-2-[(3-methyl-1-benzofuran-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
(1R,9aR)-1-[({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)methyl]-octahydro-1H-quinolizin-1-ol
N-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylcyclopropanecarbonyl)piperidine