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1-(5-chloropyridin-2-yl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
(2R,6R)-1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-2-(2-methylphenyl)-1,3-oxazole
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}-1,2,5-thiadiazole-3-carboxamide
1-(1,4-dithiepan-6-yl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-{1-[(2R)-oxolan-2-ylmethyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]benzonitrile
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbenzamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(oxolane-2-carbonyl)piperidin-4-amine
[(3R,4R)-1-(4-fluoro-3-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-(cyclopentylamino)-1-(3-phenylpropyl)pyrrolidin-2-one
[1-({methyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)cyclopropyl]methanol
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-9,10-dihydroacridin-9-one
6-(3-methylphenyl)-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carboxylic acid
5-(4-benzoylpiperidine-1-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-cyclopentanecarbonyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
8-(3-chloropyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 4-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-oxobutanoate
N-[2-(diethylamino)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-N-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)oxolan-3-amine
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxy-5-methylbenzamide
5-[4-(3-methylphenoxy)piperidine-1-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
6-(4-butylphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-cyclohexyl-3-methyl-5-[2-(1H-1,2,4-triazol-3-yl)phenyl]-1H-1,2,4-triazole
methyl 2-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
1-[3-(oxan-4-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]-6-azaspiro[2.5]octane
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
9-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-cyclopentyl-6-[4-(2-methoxyethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
ethyl 1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazole-2-carboxylate
1-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(2-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(4,5-dichloro-2-methyl-1H-imidazol-1-yl)acetamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
2-[4-(hydroxymethyl)phenyl]-1-[4-(2-methylphenoxy)piperidin-1-yl]ethan-1-one
6-[3-(1-methoxyethyl)phenyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-3-(1H-pyrazol-4-yl)propanamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-(3-fluorophenyl)-5-(3-methylbut-2-en-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(benzylsulfamoyl)({[2-(1H-pyrazol-1-yl)phenyl]methyl})amine
2-methoxy-N-(2-methoxy-5-{[methyl(1,3-thiazol-2-ylmethyl)carbamoyl]amino}phenyl)acetamide
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-{4-[({6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}amino)methyl]piperidin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
2-[2-oxo-4-(4-phenoxybutyl)piperazin-1-yl]benzonitrile
N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
(2S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-hydroxypropanamide
2-[(3-propoxypiperidin-1-yl)methyl]-1H-1,3-benzodiazole