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5-ethyl-2-methyl-4-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyrimidine
3-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
2-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2,8-dimethylquinoline
(2E)-1-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(pyridin-4-yl)prop-2-en-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
N-{[3-methoxy-4-(pyridin-2-ylmethoxy)phenyl]methyl}-N-(oxolan-2-ylmethyl)-2-(trifluoromethyl)benzamide
5-(3-acetylphenoxymethyl)-N-(3-hydroxybutyl)-1,2-oxazole-3-carboxamide
10-methoxy-5-[5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(thiophen-3-yl)propanamide
(4aS,7aR)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-N-cyclopentylpropanamide
3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
4,5-dimethyl-2-[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
9-cyclobutanecarbonyl-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]piperidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-N-methylpiperidin-4-amine
1-(furan-2-ylmethyl)-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
(2R,6R)-1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-propylacetamide
3-(3-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}butyl)-1H-indole
3-{5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(2-hydroxyethyl)propanamide
4-{[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}benzene-1-sulfonamide
1-[2-({2,7-dimethylimidazo[1,2-a]pyridin-3-yl}formamido)ethyl]piperidine-3-carboxamide
7-(1-propyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-ethoxy-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
(3aR,6aR)-2-methanesulfonyl-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-[4-(pyrimidin-4-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
5-({4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)-1-methylpiperidin-2-one
3-(piperidin-3-yl)-N-[2-(pyridin-3-yl)ethyl]benzamide
4-(pyridin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrimidin-2-amine
1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-phenylpiperidine
4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
[(3R,4R)-1-(2-methoxy-4-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-{2-[4-(2-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
(2S,4R)-4-{4-[4-(2,5-dihydro-1H-pyrrol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
(2S,4S,5R)-4-[(furan-2-ylmethyl)(methyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(2-methylphenyl)pyrrolidin-3-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-(2-methoxyphenyl)-3-{1-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridin-2-amine
(4aR,7aS)-1-(2-methylpropanoyl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-(3,4-difluorophenyl)piperidin-3-amine
1-(5-chloro-2-fluorobenzoyl)-4-cyclohexyl-1,4-diazepane
5-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-4-phenylpyrimidin-2-amine
5-methyl-3-[4-(trifluoromethyl)pyrimidin-2-yl]-1H-indole
(4aR,7aS)-1-acetyl-4-[(3-methylquinoxalin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-chloro-N,5-dimethyl-N-(quinolin-3-ylmethyl)benzamide
2-(4-ethylpiperazin-1-yl)-1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
N-ethyl-2-{4-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]piperazin-1-yl}acetamide