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8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(3-hydroxypiperidin-1-yl)sulfonyl]-N-(2,2,2-trifluoroethyl)benzamide
N-(diphenylmethyl)-2-{[2-(1-methyl-1H-imidazol-2-yl)phenyl]formamido}acetamide
6-fluoro-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4R)-N-(3-cyanophenyl)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carboxamide
N-(2-hydroxyethyl)-1-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
5-(azepane-1-carbonyl)-N-(1H-1,3-benzodiazol-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
5-(2-methoxyphenyl)-1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(thiophen-3-yl)acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-(2-methoxyethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(trifluoromethyl)benzamide
3-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzoyl]piperidine
3-(2-methoxyphenoxy)-1-(oxolane-3-carbonyl)azetidine
4-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]thiophene-2-carboxamide
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
[(3-tert-butyl-1H-pyrazol-5-yl)methyl]({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)methylamine
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
N-(1-{4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-1-oxopentan-2-yl)acetamide
dimethyl[({1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}methyl)sulfamoyl]amine
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-1,3-benzothiazole
[(3R,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-N-(pyridin-2-ylmethyl)pyridin-2-amine
4-ethyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[4-(aminomethyl)benzoyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2-hydroxyphenyl)methyl]-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
1-ethyl-8-(1H-indol-2-ylmethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1,3-benzothiazol-2-yl)-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
(3aR,6aS)-2-(cyclopropylmethyl)-5-(2-methoxybenzoyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(cyclohex-1-en-1-ylmethyl)-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{1-[(1-methyl-1H-imidazol-2-yl)methyl]azepan-4-yl}-3,4-dihydro-2H-1-benzopyran-6-carboxamide
(3aS,7aR)-5-methyl-2-(1,2-thiazole-5-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
ethyl 4-(4-{4-[methyl(oxolan-3-yl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
1,3,5-trimethyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1H-pyrazole-4-sulfonamide
5-(methanesulfonylmethyl)-2-[2-(propan-2-yloxy)phenyl]pyridine
2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
5-ethyl-N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)-1,3-oxazole-4-carboxamide
(3aR,6aR)-N,2-dimethyl-N-(quinolin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(4aR,8aS)-6-[(2-fluoro-4-methoxyphenyl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-(1-benzylpiperidin-4-yl)-N-cyclopentylpiperidine-3-carboxamide
8-methoxy-5-[6-(methoxymethyl)pyrimidin-4-yl]quinoline
N-(1,1-dioxo-1λ6-thiolan-3-yl)-6-methyl-N-(prop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3,3-dimethylbutan-1-one
9-(2-butoxyacetyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
6-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-[4-(1H-pyrazol-3-yl)benzoyl]morpholine
(4aS,7aR)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-N-[(2-fluorophenyl)methyl]-2-methanesulfonamidopropanamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide