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(4aS,8aR)-6-(1,3-benzoxazol-2-yl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]thiomorpholine
2-[4-(2-methylpyrimidine-5-carbonyl)piperazin-1-yl]-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)amine
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[4-(4-fluoro-3-methoxyphenyl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]propanamide
4-{[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}pyridin-2-ol
5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]isoquinoline
N,N-dimethyl-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(1S,6R)-3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]piperidin-3-ol
4-(6-methyl-2-propylpyrimidin-4-yl)-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
3-(2-methoxyethyl)-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
6-(benzyloxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(1H-indol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-4-(piperidin-1-yl)piperidine-4-carboxamide
3-{[cyclopropyl(1,3-thiazol-2-ylmethyl)amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
N-[(3S,4R)-4-propyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-yl]methanesulfonamide
9-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-methylpiperidin-1-yl)-2-[4-(thiomorpholin-4-ylmethyl)phenoxy]ethan-1-one
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-ethoxyethan-1-one
5-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methoxyphenol
1-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
ethyl 2-chloro-5-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}amino)benzoate
2-methyl-4-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,3-thiazole-5-carboxamide
1-(piperidin-1-yl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]cyclohexane-1-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-(3-methyloxetane-3-carbonyl)pyrrolidine-3-carboxylic acid
methyl 1-(cyclopropylmethyl)-3-[2-(1,4-diazepan-1-yl)-2-oxoethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
2-(3-methoxypropyl)-8-[2-(methylsulfanyl)pyridine-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
2-[5-(2,6-dimethoxyphenyl)-1H-indazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
dimethyl[(4-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}phenyl)methyl]amine
8-(2-hydroxyacetyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-{5-[2-(ethanesulfonyl)propanamido]-2-methoxyphenyl}furan-2-carboxamide
N4-ethyl-N2-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-2,4-diamine
8-{[4-(4-chlorophenoxy)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-1,3-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-1H-pyrazole-5-carboxamide
1-(1-benzofuran-2-ylmethyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-({4-[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}methyl)pyridine
N-[2-(3-chlorophenyl)ethyl]-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(2-methoxyphenyl)acetamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-methylpropyl)piperidine-3-carboxamide
N-[2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-4-propylpyrimidine-5-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
5-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1H-1,2,4-triazol-3-amine
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
6-[(diethylamino)methyl]-N-methyl-N-(oxan-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-cyclohexyl-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-N-methylpyridin-2-amine