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2-(ethylamino)-N-{[1-(4-fluorophenyl)cyclopentyl]methyl}pyrimidine-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(3-fluorophenyl)methyl]-3-(5-oxo-1-phenylpyrrolidin-3-yl)urea
6-{2,7-diazaspiro[4.5]decane-2-sulfonyl}-2H-chromen-2-one
5-benzyl-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-phenyl-1H-1,2,3,4-tetrazol-5-amine
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-[2-(dimethylamino)ethyl]-2-(methylamino)-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
3-hydroxy-3-{[methyl(propyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
4-chloro-1-methyl-3-{[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1H-indazole
(3R,9aR)-8-[(3-fluorophenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(butan-2-yl)-4-[5-(2-methylbenzamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
3-amino-N-[4-(4-methoxyphenoxy)phenyl]piperidine-1-carboxamide
2-cyclopentyl-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-({1-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)-5-methyl-1H-1,2,3,4-tetrazole
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(azepan-1-yl)-3-[3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-{3-[({1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}amino)methyl]-1H-indol-1-yl}propanamide
4-[(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)methyl]morpholine
1-(benzyloxy)-8-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
4-(3-hydroxy-4-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
methyl 4-{[3-ethyl-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
2-methyl-4-(2-methylphenyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperazine
2-[5-(3-cyclopentyl-1-ethyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-3-yl]pyridine
3-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-6-methyl-1-[(2-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
methyl 7-oxo-3-(1,2,5-thiadiazole-3-carbonyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)-N-methylacetamide
2-methoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pyridine-4-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(2E)-3-phenylprop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
4-(2-methyl-4-phenylpyridine-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
1-(3,3-diphenylpiperidin-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N4-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
N-methyl-3-[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
2-ethyl-N-[3-(phenylsulfanyl)propyl]pyrimidine-5-carboxamide
5-(2-methylpiperidine-1-carbonyl)-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-chlorobenzamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)propanamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine
N-[2-(3-methoxyphenyl)ethyl]-5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-amine
1-[1'-(2-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-cyclopropyl-2-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}pyridine-4-carboxamide
5-(1-butyl-1H-1,2,4-triazol-5-yl)-2-(methylsulfanyl)pyrimidine
N-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
1-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(pyridin-4-yl)propan-1-one
3-(1H-imidazol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
1-[(2,3-difluorophenyl)methyl]-4-[1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]piperidine
4-(2-{1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}ethyl)morpholine
N-methyl-2-[5-oxo-4-(2-phenylethyl)-3-(thiophen-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide