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6-oxo-1-(2-phenylethyl)-N-propyl-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-(5-oxopyrrolidin-2-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
2-[3-(4-fluorophenoxy)propyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
3-cyclobutyl-4-(3-ethoxy-2-hydroxyphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
5,7-dimethoxy-4-(8-methylquinolin-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
1-cycloheptyl-N-(2,3-dihydro-1H-inden-2-yl)-6-oxopiperidine-3-carboxamide
1-{3-[2-(azetidin-1-ylmethyl)-4-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-ethylpyrimidine-5-carboxamide
3-{[1-(2,3-dimethylphenyl)piperidin-4-yl](methyl)amino}-N-methylpropanamide
(4aR,8aS)-1-[2-(4-chloro-2-methylphenoxy)propanoyl]-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
(3aR,5S,6S,7aS)-2-[(3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-isoindole-5,6-diol
N-(3-cyanophenyl)-4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
2-(2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
1-[(3-fluorophenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
1-ethyl-4-(5-methyl-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)piperazine
1-ethyl-3-phenyl-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol
2-(2-hydroxyethyl)-8-[2-(4-methoxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3-chlorobenzoyl)-1-(2,4-difluorobenzenesulfonyl)piperidine
[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
1-(oxan-4-yl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
5-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
2-(3,4-dichlorophenyl)-6-(1-methylpiperidin-3-yl)-3,4-dihydropyrimidin-4-one
4-(1-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
4-(2-methyl-1H-imidazol-1-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}butan-1-one
4-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-2-ethyl-3-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{2-[({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]ethyl}acetamide
1-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]-3,3-dimethylbutan-1-one
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
(1S,6R)-N-[2-(3-methoxyphenyl)phenyl]-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-{[4-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-4-ol
3-[3-(2-oxopyrrolidin-1-yl)phenyl]-1-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
{1-ethyl-5-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
2-{5-[6-amino-5-cyano-4-(3-methoxyphenyl)pyridin-2-yl]thiophen-3-yl}acetic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-ethyl-N-methyl-3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-sulfonamide
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine
3-(5-chloro-1-methyl-4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-3-yl)-5-methyl-1,2-oxazole
5-methyl-3-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
2-methanesulfonamido-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
8-[(2S)-2-aminobutanoyl]-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-ethyl-3-(piperidin-4-ylmethyl)-1-(1,3-thiazol-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{3-[(4-methylphenyl)sulfanyl]propyl}acetamide
S-{4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]phenyl}-3-hydroxypropane-1-sulfonamido
4-{4-[(2-ethoxyphenyl)methyl]piperazin-1-yl}-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one