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(3aS,6aR)-5-(5-acetylpyridin-2-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[1-(2,5-dimethylphenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]pyrazin-2-ol
N-[3-(3,5-dimethylphenoxy)propyl]-N,2,4-trimethyl-1,3-oxazole-5-carboxamide
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(propan-2-yloxy)ethyl]pyrimidin-2-amine
(1S,5R)-6-[2-(methylsulfanyl)benzoyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}naphthalen-2-ol
2-({[(3-fluorophenyl)carbamoyl]amino}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(1,3-thiazol-2-yl)piperidin-4-yl]oxy}benzamide
2-methoxy-3-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)pyridine
(4aS,7aR)-1-[(2,5-difluorophenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-9-(furan-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
3-(2-amino-1,3-thiazol-4-yl)-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)propanamide
6-[(diethylamino)methyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(adamantan-1-ylmethyl)-N-methyl-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
N-(4-methoxy-2-methylphenyl)-3-(2-methoxyphenoxy)azetidine-1-carboxamide
1-ethyl-N-(furan-2-ylmethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[(2S,4S)-4-fluoro-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidin-2-yl]methyl}acetamide
(2E)-1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(thiophen-2-yl)prop-2-en-1-one
7-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](methyl){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
(2S,4R)-4-amino-N-ethyl-1-[3-methyl-4-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-(5-methoxyfuran-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
6-fluoro-8-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}quinoline
N-[3-(morpholin-4-yl)propyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2-methylphenyl)-3-{1-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
8-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]quinoline
N-(propan-2-yl)-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
(1S,5R)-3-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-(2-methylpropyl)-N-[2-(pyridin-2-yl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4-benzyl-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-4-yl)methanol
1-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(cyclohex-3-ene-1-carbonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
2-ethyl-1-(propan-2-yl)-4-(3-propyl-1H-pyrazole-4-carbonyl)piperazine
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(3,6-dimethylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
2-(1H-1,3-benzodiazol-1-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}piperidine-4-carboxamide
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-fluoropiperidine
(2R,3R)-3-(4-hydroxy-4-phenylpiperidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-methyl-5-(5-methyl-2-phenylfuran-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[methyl(quinolin-3-ylmethyl)amino]methyl}benzene-1,2-diol
(1S,5R)-3-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]propanamide