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8-(3-methylpyrazin-2-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)phenyl]pyrrolidin-2-one
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-5-methoxyfuran-2-carboxamide
N-[(3S,4R)-1-[2-(2-methyl-1H-indol-3-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-chloro-5-(3-ethoxyphenyl)pyrazine
N-(cyclohex-1-en-1-ylmethyl)-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
2-acetamido-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
(2S,4S)-N-ethyl-1-[(3-fluorophenyl)methyl]-4-[2-(1H-imidazol-1-yl)acetamido]pyrrolidine-2-carboxamide
(1R,5S)-6-methyl-3-[2-(3,4,5-trimethoxyphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-yl}pyrrolidin-3-ol
N-{4-[2-amino-3-cyano-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]phenyl}acetamide
3-{1-[3-(3-hydroxy-3-methylbutyl)phenyl]-N-methylformamido}propanamide
N-cyclopentyl-N'-[(1R)-1-(3-methoxyphenyl)ethyl]butanediamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-methylurea
4-{1-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-1,2,3-triazol-4-yl}quinoline
6-(2-methoxypyridin-3-yl)pyridine-3-carboxamide
(2S,4S,5R)-4-[(2-hydroxyethyl)(methyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
N-ethyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-methyl-N-(oxolan-2-ylmethyl)-1,2,3-thiadiazole-5-carboxamide
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)(1,2-oxazol-3-ylmethyl)amine
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
N-cyclohexyl-N-methyl-2-[(prop-2-en-1-yl)amino]benzamide
1-(1,3-benzothiazol-2-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-methoxyphenyl)propan-1-one
5-acetyl-N-[(2-ethoxyphenyl)methyl]-N-ethylthiophene-2-carboxamide
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
4-(hydroxymethyl)-1-[2-(phenylamino)pyrimidine-5-carbonyl]azepan-4-ol
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
3-methyl-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-(cyclopropylmethyl)-8-(6-phenylpyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,5S)-1-cyclopentyl-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-2-ethylpyridine-4-carboxamide
3-{4-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}phenol
4-(3-methyl-1,2,4-oxadiazol-5-yl)-1-[4-(propan-2-yl)phenyl]pyrrolidin-2-one
N,8-dimethyl-N-(1-methylpyrrolidin-3-yl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
1-cyclopentyl-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
3-methoxy-1-(2-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
N-[2-(4-methoxyphenyl)phenyl]-1-(propane-1-sulfonyl)pyrrolidine-2-carboxamide
1-[5-(2-chlorophenyl)furan-2-carbonyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
N-methyl-5-{[(3R,4S)-3-[2-(methylsulfanyl)acetamido]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}furan-2-carboxamide
3-[(4aR,7aS)-4-[(5-methylthiophen-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
5-methyl-1-(4-methylphenyl)-4-(quinoline-3-carbonyl)piperazin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-3-ol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(3-methylbutan-2-yl)-1,2-oxazole-3-carboxamide
2-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-[(pyridin-3-ylmethyl)amino]benzamide
4-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1-methylpiperazin-2-one
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N'-(2,4-dimethylphenyl)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]ethanediamide
2-amino-6-cyclobutyl-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile