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2-{4-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]morpholin-3-yl}-N-phenylacetamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
(2S,4S)-4-amino-1-(3,5-dichloro-2-hydroxybenzenesulfonyl)-N-methylpyrrolidine-2-carboxamide
(2S)-N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2,3,5-trimethyl-N-(thiolan-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-3-[(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
methyl({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)[2-(methylamino)ethyl]amine
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
5-hydroxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)pyrazine-2-carboxamide
N-(3-hydroxypropyl)-1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-(2-chloro-6-methylphenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4S)-1-(2-aminopyridine-4-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-(2-methanesulfonylethyl)-N-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
N-[(1-hydroxycyclohexyl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methylpyrazine-2-carboxamide
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropan-1-amine
2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-N-[1-(1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
3-[(butan-2-yl)amino]-N-(naphthalen-1-yl)propanamide
1-{1-[(3-cyanophenyl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-3-carboxamide
6-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)-2-methyl-2,3-dihydropyridazin-3-one
4-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
N-(2-hydroxyethyl)-5-[2-(methylsulfanyl)phenoxymethyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
8-[(6-methoxy-2H-chromen-3-yl)methyl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
methyl 5-(4-{2-[(3-methylphenyl)carbamoyl]ethyl}piperidin-1-yl)-5-oxopentanoate
N-{[(3S,4S)-3-hydroxy-1-[2-(methylsulfanyl)acetyl]piperidin-4-yl]methyl}naphthalene-1-carboxamide
1-methyl-3-(pyridin-3-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{1-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-benzyl-N-methyl-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}imidazo[1,2-a]pyridine-2-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-2-(2-oxopiperidin-1-yl)acetamide
(2,1,3-benzoxadiazol-4-ylmethyl)({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-hydroxy-3-methylbenzamide
2-[1-(thian-4-yl)pyrrolidin-2-yl]pyridine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-(1-propylpiperidin-4-yl)acetamide
5-(1H-indol-2-ylmethyl)-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
(2S,4S,5R)-4-(cyclohexylcarbamoyl)-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
4-(4-methoxyphenoxy)-1-(1H-pyrrole-2-carbonyl)piperidine
[2-(dimethylamino)ethyl]({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
5-(2,6-difluorophenoxymethyl)-N-(furan-3-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-(1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
(4aR,8aR)-2-methanesulfonyl-7-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
1-(cyclopropanesulfonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}propanamide
4,6-dimethyl-3-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-4-propyl-1,4-diazepan-5-one
N,1-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(phenylamino)pyrimidine-5-carboxamide
2-{2-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one