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(1R,9aR)-1-({4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-octahydro-1H-quinolizin-1-ol
[1-(2-aminopyrimidin-4-yl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
2-(4-fluorophenoxymethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]propanamide
6-fluoro-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(cyclohexylmethyl)-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
5-hydroxy-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrazine-2-carboxamide
1-benzoyl-4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]-3-phenylpropanoic acid
1-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-[2-(trifluoromethyl)phenyl]-1H-imidazole
1-(1,3-dihydro-2-benzofuran-5-yl)-3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
6-ethoxy-3-[(3-oxo-1,4-diazepan-1-yl)methyl]-1,2-dihydroquinolin-2-one
N-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}methanesulfonamide
(3aR,6aR)-2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-methyl-1-propyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl][(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]methylamine
8-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-1-oxa-8-azaspiro[4.5]decan-3-ol
1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(hydroxymethyl)azepan-4-ol
1-benzyl-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
3-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-1-[(2-methylpyridin-4-yl)methyl]urea
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
(3R)-1-({5-[(2,3-difluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methylpiperazine
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-1-(2H-1,3-benzodioxol-5-ylmethyl)-3-phenylpyrrolidine-2,5-dione
2-({[(3R,4R)-4-(hydroxymethyl)-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-methyl-4-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propoxy}piperidine
N-[(3-chlorophenyl)methyl]-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]propanamide
N-benzyl-N-(cyclobutylmethyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
methyl({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})[2-(methylsulfanyl)ethyl]amine
N-[(3-methoxyphenyl)methyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-(2-methylpropyl)propanamide
N-[(4-methyl-1,4-oxazepan-6-yl)methyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
5-acetyl-N-[3-(cyclohexyloxy)propyl]thiophene-3-carboxamide
N-benzyl-N-cyclopentyl-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-[(4-chlorophenyl)methyl]-6-oxo-N-[(1r,4r)-4-hydroxycyclohexyl]piperidine-3-carboxamide
(5S)-5-({[(5-cyclohexylthiophen-2-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-N-(3-fluorophenyl)-2-oxoacetamide
2-(4-{[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-yl)pyrazine
N-cyclopropyl-4-hydroxy-N-[(3-hydroxyphenyl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
{1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylacetamide
1-[2-(1H-imidazol-1-yl)ethyl]-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-[(2R,3R)-2-methoxy-1'-(5-methylpyrazine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
[2-({4-[(2,6-difluorophenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-4-[2-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-4-(2,2-dimethyloxan-4-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-{2-[1-(4-fluorophenyl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
9-(2-methyl-1H-pyrrole-3-carbonyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
1-cyclohexyl-N3-methyl-N5-(2-methylpropyl)-4-oxo-N3-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide