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1-(2,3-dihydro-1H-inden-2-yl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-diazepane
1-ethyl-6-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]piperidine-3-carboxamide
6-(4-chlorophenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-2,6-dimethylquinoline-3-carboxamide
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(3,4-difluorophenyl)propanamide
(2S)-2-{[3-(4-fluorophenyl)-1H-pyrazol-5-yl]formamido}-3-(1H-imidazol-4-yl)propanamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-(cyclopropylmethyl)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-ethyl-1-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indazole-3-carboxamide
1-(3,5-difluorophenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
3-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
2-(2-{1-[4-(trifluoromethyl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-[2-(pyridin-2-ylsulfanyl)ethyl]oxane-2-carboxamide
1-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-3-(oxolan-2-ylmethyl)-3-propylurea
2-(4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}phenoxymethyl)pyridine
3-chloro-4-fluoro-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-1-benzothiophene-2-carboxamide
3-{[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}propane-1,2-diol
2-phenyl-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-methoxy-2-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]methyl}phenol
3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1-{[1-(morpholin-4-yl)cyclohexyl]methyl}urea
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)propanamide
1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
N-{1-[(5-phenylthiophen-2-yl)methyl]piperidin-4-yl}methanesulfonamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
3-(5-methyl-1,2,4-oxadiazol-3-yl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide
2-(benzylsulfamoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
6-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-2-methylpyrimidin-4-ol
N-ethyl-1-methyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
N3-benzyl-N5-[2-(3-fluorophenyl)ethyl]-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(methoxymethyl)-5-(2-phenyl-1H-imidazol-4-yl)-1,2,4-oxadiazole
(3R,4R)-4-(morpholin-4-yl)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-ol
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
7-(cyclopropylmethyl)-2-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
[2-(2-ethylphenoxy)ethyl]({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})methylamine
1-(2-aminoethyl)-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(4-chloro-3-methylphenyl)-2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)acetamide
(1R,5R)-3-methanesulfonyl-6-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carboxamide
{5-[1-(2,2,6-trimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-1H-imidazol-2-yl]furan-2-yl}methanol
N-(butan-2-yl)-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-(pyridin-3-ylmethyl)propanamide
(4R)-1-(3-benzyl-1,2,4-oxadiazol-5-yl)-4,7,7-trimethyl-2-oxabicyclo[2.2.1]heptan-3-one
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-2-one
N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-4-(trifluoromethyl)pyrimidin-2-amine
(3-{2-[1-(3,4-dimethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
4-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
methyl 1-oxo-2-({5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-1,2-dihydroisoquinoline-7-carboxylate