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1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(1-methyl-1H-1,2,3-triazol-4-yl)-3-({2-[(methylcarbamoyl)methyl]-3-oxopiperazin-1-yl}methyl)benzamide
3-butyl-1-methyl-4-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperazin-2-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-hydroxy-4-methylbenzamide
N-(furan-3-ylmethyl)-N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
(3-propyl-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl)methanol
(2S,4S)-4-amino-1-[2-(4-cyclopropaneamidophenyl)acetyl]-N-methylpyrrolidine-2-carboxamide
N-(3-chloro-2-methylphenyl)-3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carboxamide
2-(carbamoylamino)-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]urea
7-(cyclohexylmethyl)-2-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-2,7-diazaspiro[4.5]decane
4-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}benzamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]acetamide
2-[4-(dimethylamino)phenyl]-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]ethan-1-one
3,6-dimethyl-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-{[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}-1-(propan-2-yl)pyrrolidin-2-one
N4-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-4,6-diamine
7-(5-methylthiophen-2-yl)-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(butane-1-sulfonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}thiophen-2-yl)ethan-1-one
4-(4-fluorophenoxy)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidine
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}propanamide
(1S,5R)-3-acetyl-N-(5-chloro-2-methylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-N-(propan-2-yl)pyrimidin-2-amine
1-{2-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
N-(2,3-dihydroxypropyl)-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
methyl 5-[2-(pyridin-4-ylsulfanyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-(4-{[methyl(thian-4-yl)amino]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
8-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-4-phenylbutan-1-one
methyl 1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
3-cyclohexyl-4-(dimethyl-1,2-oxazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(5-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-1H-pyrazol-3-yl)phenol
{5-methyl-7-[3-(trifluoromethyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-({[(3R,4R)-4-(hydroxymethyl)-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
({5-[(3-benzoylpiperidin-1-yl)methyl]thiophen-3-yl}methyl)dimethylamine
4-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
4-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}thiomorpholine
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-(pyrrolidine-1-carbonyl)piperazine
(2R,6S)-1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(propan-2-yloxy)ethan-1-one
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
2-(2-{4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
7-fluoro-2-methyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-4-carboxamide
2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
2-{3-[1-(2-ethoxyethyl)-1H-pyrazol-3-yl]phenyl}-4,6-dimethylpyrimidine
(1R,5S,6S)-6-({4-[(2-methoxyphenyl)methyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
N-cyclopentyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)propanamide