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3-[3-({[1-(3-fluoro-4-methoxyphenyl)ethyl]carbamoyl}amino)phenyl]-N-methylpropanamide
2-[3-(1H-imidazol-1-yl)propyl]-9-(propane-2-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3-fluoro-4-methoxyphenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
3-(4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}piperidine-1-carbonyl)pyridine
ethyl 2-{1-[(2-fluorophenyl)methanesulfonyl]piperidin-2-yl}acetate
methyl 4-{[5-(2,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}butanoate
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(2-methoxyethyl)[(4-methylphenyl)methyl]{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-[(3-phenyloxolan-3-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
2-cyclopentyl-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{[(3S)-piperidin-3-yl]sulfamoyl}benzamide
4-methoxy-6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
2-(1-{1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-(1,3-oxazole-5-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[2-(2-methylbutanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
8-{imidazo[1,2-a]pyridine-2-carbonyl}-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
4-{3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}morpholine
(4aR,7aS)-1-[2-(4-ethyl-1,4-diazepan-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
1-cyclopropyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrrolidin-2-one
1-(pyrimidin-2-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-cyclopentyl-4-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]pyrrolidin-2-one
4-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}thiomorpholine
5-methyl-2-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}pyrimidin-4-amine
3-(2-phenylethyl)-5-[5-(thiophen-2-yl)-1H-pyrazol-4-yl]-1H-1,2,4-triazole
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine-3-carboxamide
2-(4-fluorophenyl)-2-hydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
4-({4-methyl-5-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-(2H-1,3-benzodioxol-5-yl)-N-{[7-(4-cyclopropanecarbonylphenyl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
1-(2-methoxyphenyl)-2,2-dimethyl-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
N-methyl-5-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2-methoxyphenol
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
1-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-4-methoxy-4-(prop-2-en-1-yl)piperidine
2-(3-{3-[cyclohexyl(methyl)amino]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)-N-ethylacetamide
(3R)-1-[(1-{[1-(4,5-dimethylthiophene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-amine
methyl 3-benzamido-6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
5-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidine
5-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-N-ethylpyrimidin-2-amine
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-(3-cyanothiophen-2-yl)-4-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)benzamide
2-{[4-(3-methoxyphenyl)-5-(1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-benzyl-8-[(3-methylthiophen-2-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
7-(3-chlorophenyl)-4-cyclobutanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-hydroxyphenyl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
3-(3-fluoro-4-phenylbenzoyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,2-dihydroquinolin-2-one