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N-cyclopentyl-4-acetamido-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzamide
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(4-methylphenyl)propanamide
1-(5-fluoro-2-methylbenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
4-chloro-1-methyl-3-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}-1H-indazole
4-phenoxy-1-[(2E)-3-phenylprop-2-enoyl]piperidine-4-carboxylic acid
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
N-(pyridin-3-ylmethyl)-4-{4-[(thiophen-2-ylmethyl)amino]piperidin-1-yl}benzamide
3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-[(5-methylthiophen-2-yl)methyl]benzamide
2-amino-4-(3-chloro-4-hydroxy-5-methoxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-methyl-4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-cyclopropyl-1-(2,6-dimethoxypyridin-3-yl)-3-(thiophen-3-ylmethyl)urea
4-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}thiomorpholine
4-{3-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]butyl}phenol
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
5-methyl-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(8-chloroquinolin-2-yl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylic acid
2-[(3R,4R)-3-hydroxy-4-(morpholin-4-yl)piperidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
3-[(5-methyl-4-phenyl-1H-imidazol-1-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridin-2-amine
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1,5-dimethyl-4-{[methyl(thian-4-yl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(3S,4R)-4-(3-methoxyphenyl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
(4aS,8aR)-1-(3-hydroxypropyl)-6-(pyrimidine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(3-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyridin-2-yl)-2,2-dimethylpropanamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-benzoyl-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
(1,4-dioxan-2-ylmethyl)(methyl){[5-(2-methylpropyl)thiophen-2-yl]methyl}amine
N-(3-fluorophenyl)-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydroquinoxalin-2-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
1-{1-[(4-fluoro-3-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
4-benzyl-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-ol
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
ethyl 1-[(3,4-dimethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
2-({[(3R,4R)-1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-2-carbonitrile
3-[2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]-1,3-oxazinan-2-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-methyl-N-(oxolan-2-ylmethyl)benzamide
2-(3,4-dichlorophenyl)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]morpholine
2-methyl-4-phenyl-9-[2-(propan-2-ylsulfanyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{imidazo[1,2-a]pyridin-2-yl}-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
7,7-dimethyl-2-[2-(2-methyl-1H-imidazol-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{1-[(5-ethylfuran-2-yl)methyl]piperidin-2-yl}ethyl)-4-methylpiperazine
methyl 1-ethoxy-8-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(3aS,6aR)-5-(4,6-dimethylpyrimidin-2-yl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one