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2-{4-[3-(difluoromethoxy)benzoyl]-2-oxopiperazin-1-yl}benzonitrile
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(2-chlorophenyl)-2-hydroxy-1-{4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
N-[2-(1,3-benzoxazol-2-yl)ethyl]-4-sulfamoylbenzamide
N-methyl-3-(5-methylthiophen-2-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
N,N-dimethyl-5-[4-(thian-4-yl)piperazine-1-carbonyl]pyridin-2-amine
N-[(4-fluorophenyl)methyl]-3-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]propanamide
2-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
4-(4-methoxyphenoxy)-1-(1-methylpiperidine-2-carbonyl)piperidine
6-methyl-3-[4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
N-cyclopropyl-1-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]piperidine-4-carboxamide
(4aS,8aR)-6-[2-(2,4-dimethylphenoxy)ethyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-3-hydroxypropanoic acid
N-(1-hydroxypropan-2-yl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
3-amino-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-1,2,4-triazole-5-carboxamide
ethyl 4-benzyl-1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidine-4-carboxylate
2-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}quinoline
(3S,4S)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
(3aR,6aR)-2-methanesulfonyl-5-(3-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-4-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydroquinoline-2-carboxamide
4-{[7-(3-methylbut-2-en-1-yl)-3-(oxan-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-5-yl]methyl}-1H-imidazole
4-{[(2E)-2-methylbut-2-en-1-yl]amino}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2-(2-chlorophenyl)morpholin-4-yl]ethan-1-one
(2S,4R)-1-benzyl-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
1-phenyl-3-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]pyrrolidin-2-one
4-[2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carbonyl]thiomorpholine
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
N,N-diethyl-2-[4-(3-propyl-1,2,4-oxadiazol-5-yl)-1H-1,2,3-triazol-1-yl]acetamide
6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
(3R,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-methyl-5-{5-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
methyl 3-(2-chlorobenzamido)-5-({[3-(dimethylamino)phenyl]formamido}methyl)benzoate
N-(5-chloro-2-methoxyphenyl)-3-[1-(2-cyclopentylacetyl)piperidin-3-yl]propanamide
methyl[1-(1,2-oxazol-3-yl)ethyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-(2,4-difluorophenyl)-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
2-{2-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(2-{[(3R)-3-methylpiperazin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)ethan-1-one
[(4-{2-[4-(furan-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
(2E)-N-{[1-(but-2-yn-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-N-methyl-3-phenylprop-2-enamide
2-(2-{[(2-chlorophenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-(3-chloro-4-hydroxyphenyl)-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
N-(3-benzylphenyl)-3-cyanopiperidine-1-carboxamide
(2S)-2-[(4-tert-butylcyclohexyl)amino]-3-methylbutan-1-ol
3-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,4S)-5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl 1-[5-(benzylcarbamoyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carbonyl]piperidine-2-carboxylate