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2-[3-(dimethylamino)pyrrolidin-1-yl]-N-[3-(2-phenylacetamido)phenyl]acetamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]propan-1-one
[(3S,5R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-({1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperidin-3-ol
N-ethyl-2,2-dimethyl-N-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)oxan-4-amine
N-(pyridin-3-yl)-5-(pyrimidin-5-yl)furan-2-carboxamide
methyl 3-[6-(trifluoromethyl)pyridin-2-yl]benzoate
1-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
4-methyl-1-(5-methyl-1H-indole-2-carbonyl)-1,4-diazepan-5-one
5-chloro-2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
2-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-[(3S,4R)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-N-methyl-N-phenylacetamide
2-(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
[1-({1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
(2R)-2-cyclohexyl-2-hydroxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
3-ethyl-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(pyrazin-2-yl)-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}phenol
1-(2-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-(dimethylamino)-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-methylpyrimidine-5-carboxamide
3-cyclopropyl-3-[(5-methylthiophen-2-yl)methyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
2-propyl-8-(3-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]phenyl}phenol
7-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{4-[6-amino-5-cyano-4-(4-hydroxy-3-methylphenyl)pyridin-2-yl]phenoxy}acetic acid
2-hydroxy-5-{[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]methyl}benzoic acid
3-cyano-5-fluoro-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)benzamide
(4aR,8aS)-1-butyl-6-[(4-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
(1R,3S)-7-(2-phenylethyl)-7-azaspiro[3.5]nonane-1,3-diol
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
3-(3-methylphenoxymethyl)-N-(pyridin-3-yl)piperidine-1-carboxamide
(1S,6R)-3-{[2-(prop-2-yn-1-yloxy)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
4-ethyl-3-(4-hydroxy-3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(adamantan-2-ylmethyl)-6-{[(cyclopropylmethyl)(propyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(4-fluorobutyl)-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
(3R,5S)-1-benzyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-(2-phenylethyl)piperidine-3-carboxamide
N-cyclopentyl-1-methyl-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(1H-indazol-1-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
2-(cyclopropylmethyl)-9-[(3-methylpyridin-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
9-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,9-diazaspiro[5.6]dodecane
1-acetyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]piperidine-3-carboxamide
4-cyclopentyl-N-[3-(4-fluorophenyl)phenyl]-3-oxopiperazine-1-carboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}oxolane-2-carboxamide
8-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-methyl-4-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]-1,2,5-oxadiazole
[(3R,5R)-1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
1-(2-phenylphenyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}urea